Synthesis, structure and antibacterial activity of novel 1-(5-substituted-3-substituted-4,5-dihydropyrazol1-yl)ethanone oxime ester derivatives
- Author
- LIU, Xin-Hua1 ; PIN CUI1 ; SONG, Bao-An2 ; BHADURY, Pinaki S2 ; ZHU, Hai-Liang1 3 ; WANG, Shi-Fan1
[1] Key Laboratory of Anhui Educational Department, Anhui University of Technology, Maanshan 243002, China
[2] Key Laboratory of Green Pesticide and Agriculture Bioengineering, Ministry of Education, Guizhou University, Guiyang 550025, China
[3] State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University, Nanjing 210093, China - Source
Bioorganic & medicinal chemistry. 2008, Vol 16, Num 7, pp 4075-4082, 8 p ; ref : 24 ref
- ISSN
- 0968-0896
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier Science, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Author keyword
- 5-Arylpyrazole Antibacterial activity Oxime ester Synthesis
- Keyword (fr)
- Activité biologique Antibactérien DNA topoisomerase (ATP-hydrolysing) Dérivé du pyrazole Escherichia coli Ester Fluor Composé organique In vitro Oxime Staphylococcus aureus Synthèse chimique Benzoïque acide(4-trifluorométhyl) ester 1-(4,5-dihydro-5-méthoxy-3-phénylpyrazol-1-yl)éthylimino Pyrazoline dérivé Bactérie Enterobacteriaceae Enzyme Isomerases Micrococcaceae Micrococcales
- Keyword (en)
- Biological activity Antibacterial agent DNA topoisomerase (ATP-hydrolysing) Pyrazole derivatives Escherichia coli Ester Fluorine Organic compounds In vitro Oxime Staphylococcus aureus Chemical synthesis Bacteria Enterobacteriaceae Enzyme Isomerases Micrococcaceae Micrococcales
- Keyword (es)
- Actividad biológica Antibacteriano DNA topoisomerase (ATP-hydrolysing) Pirazol derivado Escherichia coli Ester Fluor Compuesto orgánico In vitro Oxima Staphylococcus aureus Síntesis química Bacteria Enterobacteriaceae Enzima Isomerases Micrococcaceae Micrococcales
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S02 Antibacterial agents
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 20272664
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmc.2008.01.035 
https://dx.doi.org/10.1016/j.bmc.2008.01.035
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