Synthesis and Evaluation of Technetium-99m-and Rhenium-Labeled Inhibitors of the Prostate-Specific Membrane Antigen (PSMA)
- Author
- BANERJEE, Sangeeta R1 ; FOSS, Catherine A1 ; CASTANARES, Mark2 ; MEASE, Ronnie C1 ; BYUN, Youngjoo1 ; FOX, James J1 ; HILTON, John1 ; LUPOLD, Shawn E3 ; KOZIKOWSKI, Alan P4 ; POMPER, Martin G1 2
[1] Russell H. Morgan Department of Radiology and Radiological Sciences, Johns Hopkins Medical Institutions, Baltimore, Maryland 21231, United States
[2] Department of Pharmacology & Molecular Sciences, Johns Hopkins Medical Institutions, Baltimore, Maryland 21231, United States
[3] Department of Urology, Johns Hopkins Medical Institutions, Baltimore, Maryland 21231, United States
[4] Department of Medicinal Chemistry and Pharmacognosy, University of Illinois, Chicago, Illinois 60612, United States - Source
Journal of medicinal chemistry (Print). 2008, Vol 51, Num 15, pp 4504-4517, 14 p ; ref : 61 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Agent scintigraphique Animal Antigène membranaire spécifique prostate Captation Cellule tumorale Composé marqué Coordinat organique Distribution Dérivé de la pyridine Dérivé de la quinoléine Glutamate carboxypeptidase II Homme In vitro In vivo Inhibiteur Lignée cellulaire Produit diagnostic Produit radioisotopique Prostate Rhénium Carbonyle Complexe Souris Spectrométrie fluorescence Synthèse chimique Technétium Carbonyle Complexe Tissu Tomoscintigraphie émission monophotonique Urées Biodistribution Glutamique acide dérivé Hexanoïque acide dérivé Lignée PC3 Lysine dérivé Octanediamide dérivé Technétium 99m Enzyme Hydrolases Mammalia Metallocarboxypeptidases Métal transition Carbonyle Complexe Peptidases Rodentia Vertebrata
- Keyword (en)
- Biological activity Scintigraphic agent Animal Prostate specific membrane antigen Uptake Tumor cell Labelled compound Organic ligand Distribution Pyridine derivatives Quinoline derivatives Glutamate carboxypeptidase II Human In vitro In vivo Inhibitor Cell line Diagnostic agent Radioisotopic product Prostate Rhenium Carbonyl Complexes Mouse Fluorescence spectrometry Chemical synthesis Technetium Carbonyl Complexes Tissue Single photon emission tomography Ureas Enzyme Hydrolases Mammalia Metallocarboxypeptidases Transition metal Carbonyl Complexes Peptidases Rodentia Vertebrata
- Keyword (es)
- Actividad biológica Agente centelleográfico Animal Antígeno membranar específico prostata Captación Célula tumoral Compuesto marcado Ligando orgánico Distribución Piridina derivado Quinolina derivado Glutamate carboxypeptidase II Hombre In vitro In vivo Inhibidor Línea celular Producto diagnóstico Producto radioisotópico Prostata Renio Carbonilo Complejo Ratón Espectrometría fluorescencia Síntesis química Tecnecio Carbonilo Complejo Tejido Tomografía emisión fotón único Ureas Enzima Hydrolases Mammalia Metallocarboxypeptidases Metal transición Carbonilo Complejo Peptidases Rodentia Vertebrata
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02T Contrast media. Radiopharmaceuticals
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 20579675
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm800111u 
https://dx.doi.org/10.1021/jm800111u
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