Allele-specific inhibition of divergent protein tyrosine phosphatases with a single small molecule
- Author
- ZHANG, Xin-Yu1 ; CHEN, Vincent L1 ; ROSEN, Mari S1 ; BLAIR, Elizabeth R1 ; MARI LONE, Anna1 ; BISHOP, Anthony C1
[1] Amherst College, Department of Chemistry, Amherst, MA 01002, United States - Source
Bioorganic & medicinal chemistry. 2008, Vol 16, Num 17, pp 8090-8097, 8 p ; ref : 36 ref
- ISSN
- 0968-0896
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier Science, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Author keyword
- Allele-specific inhibitors FlAsH Inhibitor sensitization Protein tyrosine phosphatases
- Keyword (fr)
- Cinétique Hétérocycle soufre arsenic Inhibiteur enzyme Molécule petite Mutation Protein-tyrosine-phosphatase Sélectivité 1,3,2-Dithiaarsolane dérivé Benzoïque acide(2-[4,5-bis(1,3,2-dithiaarsolan-2-yl)-3,6-dihydroxyxanthén-9-yl]) Fluorescéine dérivé Enzyme Esterases Hydrolases Phosphoric monoester hydrolases
- Keyword (en)
- Kinetics Sulfur arsenic heterocycle Enzyme inhibitor Small molecule Mutation Protein-tyrosine-phosphatase Selectivity Enzyme Esterases Hydrolases Phosphoric monoester hydrolases
- Keyword (es)
- Cinética Heterociclo azufre arsénico Inhibidor enzima Molécula pequeña Mutación Protein-tyrosine-phosphatase Selectividad Enzima Esterases Hydrolases Phosphoric monoester hydrolases
- Classification
- Pascal
- 002 Biological and medical sciences / 002A Fundamental and applied biological sciences. Psychology / 002A02 Analytical, structural and metabolic biochemistry / 002A02E Enzymes and enzyme inhibitors / 002A02E04 Hydrolases
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02W Miscellaneous
- Discipline
- Analytical, structural and metabolic biochemistry General pharmacology
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 20667209
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmc.2008.07.053 
https://dx.doi.org/10.1016/j.bmc.2008.07.053
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