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ABCB1 Polymorphisms Influence Steady-State Plasma Levels of 9-Hydroxyrisperidone and Risperidone Active Moiety

Author
GUNES, Arzu1 ; SPINA, Edoardo2 3 ; DAHL, Marja-Liisa1 ; GABRIELLA SCORDO, Maria1
[1] Department of Medical Sciences, Clinical Pharmacology, Uppsala University, Uppsala, Sweden
[2] Department of Clinical and Experimental Medicine and Pharmacology, University of Messina, Messina, Italy
[3] IRCCS Centro Neurolesi Bonino-Pulejo,, Messina, Italy
Source

Therapeutic drug monitoring. 2008, Vol 30, Num 5, pp 628-633, 6 p ; ref : 42 ref

CODEN
TDMODV
ISSN
0163-4356
Scientific domain
Pharmacology drugs
Publisher
Lippincott Williams & Wilkins, Hagerstown, MD
Publication country
United States
Document type
Article
Language
English
Author keyword
9-hydroxyrisperidone ABCB1 CYP3A4 CYP3A5 risperidone
Keyword (fr)
Antipsychotique atypique Cytochrome P450 Génotype Isozyme Liquide biologique Pharmacocinétique Plasma sanguin Polymorphisme Rispéridone Variabilité génétique Cytochrome P450 3A4 Cytochrome P450 3A Antagoniste dopamine Antagoniste sérotonine Benzisoxazole dérivé Enzyme Neuroleptique Psychotrope Récepteur dopaminergique D2 Récepteur sérotoninergique
Keyword (en)
Atypical antipsychotic Cytochrome P450 Genotype Isozyme Biological fluid Pharmacokinetics Blood plasma Polymorphism Risperidone Genetic variability Dopamine antagonist Serotonin antagonist Benzisoxazole derivatives Enzyme Neuroleptic Psychotropic D2 Dopamine receptor Serotonine receptor
Keyword (es)
Antipsicótico atípico Citocromo P450 Genotipo Isozima Líquido biológico Farmacocinética Plasma sanguíneo Polimorfismo Risperidona Variabilidad genética Antagonista dopamina Antagonista serotonina Benzisoxazol derivado Enzima Neuroléptico Psicotropo Receptor dopaminérgico D2 Receptor serotoninérgico
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments

Discipline
General pharmacology
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
20742831

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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