Nonsteroidal Selective Androgen Receptor Modulators (SARMs): Dissociating the Anabolic and Androgenic Activities of the Androgen Receptor for Therapeutic Benefit
- Author
- MOHLER, Michael L1 ; BOHL, Casey E1 ; JONES, Amanda1 ; COSS, Christopher C1 ; NARAYANAN, Ramesh1 ; YALI HE1 ; DONG JIN HWANG1 ; DALTON, James T1 ; MILLER, Duane D1 2
[1] Preclinical Research and Development, GTx, Inc., 3 North Dunlap Street, Memphis, Tennessee 38163, United States
[2] Department of Pharmaceutical Sciences, College of Pharmacy, University of Tennessee Health Science Center, 847 Monroe Avenue, Memphis, Tennessee 38163, United States - Source
Journal of medicinal chemistry (Print). 2009, Vol 52, Num 12, pp 3597-3617, 21 p ; ref : 162 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Columbus, OH
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Affinité Agoniste Anabolisant Androgène Article synthèse Composé non stéroïde Récepteur androgène Récepteur hormonal Sarcopénie Modulateur sélectif récepteur androgène
- Keyword (en)
- Biological activity Affinity Agonist Anabolic agent Androgen Review Non steroid compound Androgen receptor Hormonal receptor Sarcopenia selective androgen receptor modulator
- Keyword (es)
- Actividad biológica Afinidad Agonista Agente anabólico Andrógeno Artículo síntesis Compuesto no esteroide Receptor andrógeno Receptor hormonal Sarcopenia
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02O Hormones. Endocrine system
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 21661016
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm900280m 
https://dx.doi.org/10.1021/jm900280m
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