Cytotoxic activity of 3-(5-phenyl-3H-[1,2,4]dithiazol-3-yl)chromen-4-ones and 4-oxo-4H-chromene-3-carbothioic acid N-phenylamides
- Author
- RAJ, Tilak1 ; RICHA KAUR BHATIA1 ; KAPUR, Ashish1 ; SHARMA, Madhunika2 ; SAXENA, A. K2 ; ISHAR, M. P. S1
[1] Bio-Organic and Photochemistry Laboratory, Department of Pharmaceutical Sciences, Guru Nanak Dev University, Amritsar 143 005, Punjab, India
[2] Pharmacology Division, Indian Institute of Integrative Medicine, Jammu 180 001, Jammu & Kashmir, India - Source
European journal of medicinal chemistry. 2010, Vol 45, Num 2, pp 790-794, 5 p ; ref : 37 ref
- CODEN
- EJMCA5
- ISSN
- 0223-5234
- Scientific domain
- Organic chemistry; Pharmacology drugs
- Publisher
- Elsevier, Kidlington
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Author keyword
- Anticancer activity Anticancer agents Chromanyldithiazoles Dithiazoles N-Phenylthioamides Topoisomerase inhibitors
- Keyword (fr)
- Anticancéreux Cellule tumorale Composé aromatique Composé bicyclique Cytotoxicité DNA topoisomerase Dérivé de la chromone Homme Hétérocycle oxygène In vitro Inhibiteur de la topoisomérase I Inhibiteur enzyme Lignée cellulaire Relation structure activité Synthèse chimique Thioamide 1,2,4-Dithiazole dérivé 1-Benzopyran-4-one dérivé 1-Benzopyrane-3-carbothioamide dérivé Enzyme Isomerases
- Keyword (en)
- Antineoplastic agent Tumor cell Aromatic compound Bicyclic compound Cytotoxicity DNA topoisomerase Chromone derivatives Human Oxygen heterocycle In vitro Topoisomerase I inhibitor Enzyme inhibitor Cell line Structure activity relation Chemical synthesis Thioamide Enzyme Isomerases
- Keyword (es)
- Anticanceroso Célula tumoral Compuesto aromático Compuesto bicíclico Citotoxicidad DNA topoisomerase Hombre Heterociclo oxígeno In vitro Inhibidor topoisomerase I Inhibidor enzima Línea celular Relación estructura actividad Síntesis química Tioamida Enzima Isomerases
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02R Antineoplastic agents / 002B02R01 General aspects
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 22383565
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.ejmech.2009.11.001 
https://dx.doi.org/10.1016/j.ejmech.2009.11.001
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