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Non-nucleoside reverse transcriptase inhibitors (NNRTIs), their discovery, development, and use in the treatment of HIV-1 infection: A review of the last 20 years (1989-2009)

Author
DE BETHUNE, Marie-Pierre1
[1] Tibotec BVBA, Generaal De Wittelaan L11 B3, 2800 Mechelen, Belgium
Issue title
Twenty-five Years of Antiretroviral Drug Development: Progress and Prospects
Author (monograph)
ESTE, José A (Editor)1 ; CIHLAR, Tomas (Editor)2
[1] Hospital Germans Trias i Pujol, Barcelona, Spain
[2] Gilead Sciences Inc., California, United States
Source

Antiviral research. 2010, Vol 85, Num 1, pp 75-90, 16 p ; ref : 4 p.3/4

CODEN
ARSRDR
ISSN
0166-3542
Scientific domain
Microbiology, infectious diseases; Pharmacology drugs; Virology
Publisher
Elsevier, Kidlington
Publication country
United Kingdom
Document type
Article
Language
English
Author keyword
Efavirenz Etravirine NNRTI Nevirapine Next generation NNRTI Rilpivirine
Keyword (fr)
Antirétroviral Antiviral Article synthèse Association médicamenteuse Composé non nucléoside Développement Efavirenz Etravirine Inhibiteur reverse transcriptase Médicament Névirapine Pharmacothérapie Revue bibliographique Rilpivirine SIDA Traitement Virus HIV1 Composé acétylénique Dérivé de la benzoxazine Enzyme Immunodéficit Immunopathologie Infection Inhibiteur allostérique Inhibiteur enzyme Lentivirus Nucleotidyltransferases RNA-directed DNA polymerase Retroviridae Transferases Virose Virus immunodéficience humaine Virus
Keyword (en)
Antiretroviral agent Antiviral Review Drug combination Non nucleoside compound Development Efavirenz Etravirine Reverse transcriptase inhibitor Drug Nevirapine Pharmacotherapy Bibliographic review Rilpivirine AIDS Treatment HIV-1 virus Acetylenic compound Benzoxazine derivatives Enzyme Immune deficiency Immunopathology Infection Allosteric inhibitor Enzyme inhibitor Lentivirus Nucleotidyltransferases RNA-directed DNA polymerase Retroviridae Transferases Viral disease Human immunodeficiency virus Virus
Keyword (es)
Antiretroviral Antiviral Artículo síntesis Asociación medicamentosa Compuesto no nucleósido Desarrollo Efavirenz Etravirina Inhibitor reverse transcriptase Medicamento Nevirapina Farmacoterapia Revista bibliográfica Rilpivirina SIDA Tratamiento HIV-1 virus Compuesto acetilénico Benzoxazina derivado Enzima Inmunodeficiencia Inmunopatología Infección Inhibidor alostérico Inhibidor enzima Lentivirus Nucleotidyltransferases RNA-directed DNA polymerase Retroviridae Transferases Virosis Human immunodeficiency virus Virus
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S05 Antiviral agents

Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B05 Infectious diseases / 002B05C Viral diseases / 002B05C02 Human viral diseases / 002B05C02D Viral diseases of the lymphoid tissue and the blood. Aids

Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B06 Immunopathology / 002B06D Immunodeficiencies. Immunoglobulinopathies / 002B06D01 Immunodeficiencies

Discipline
Immunopathology Infectious pathology Pharmacological treatments
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
22428965

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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