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Tumor selective delivery of 5-fluorouracil by capecitabine, a new oral fluoropyrimidine carbamate, in human cancer xenografts

Author
ISHIKAWA, T1 ; UTOH, M1 ; SAWADA, N1 ; NISHIDA, M1 ; FUKASE, Y1 ; SEKIGUCHI, F1 ; ISHITSUKA, H1
[1] Cytostatics Group, Nippon Roche Research Center, Kamakura-city, Kanagawa 247, Japan
Source

Biochemical pharmacology. 1998, Vol 55, Num 7, pp 1091-1097 ; ref : 11 ref

CODEN
BCPCA6
ISSN
0006-2952
Scientific domain
Biochemistry, molecular biology, biophysics; Pharmacology drugs; Physiology, morphology
Publisher
Elsevier Science, New York, NY
Publication country
United States
Document type
Article
Language
English
Keyword (fr)
Activité biologique Animal Anticancéreux Capécitabine Cellule tumorale Chimiothérapie Fluoropyrimidine dérivé Fluorouracil Homme Hétérogreffe Lignée cellulaire établie Métabolite Pharmacocinétique Promédicament Souris Toxicité Traitement Tumeur maligne Voie intrapéritonéale Voie orale Mammalia Rodentia Vertebrata
Keyword (en)
Biological activity Animal Antineoplastic agent Capecitabine Tumor cell Chemotherapy Fluoropyrimidine derivatives Fluorouracil Human Heterograft Established cell line Metabolite Pharmacokinetics Prodrug Mouse Toxicity Treatment Malignant tumor Intraperitoneal administration Oral administration Mammalia Rodentia Vertebrata
Keyword (es)
Actividad biológica Animal Anticanceroso Capecitabina Célula tumoral Quimioterapia Fluoropirimidina derivado Fluorouracilo Hombre Heteroinjerto Línea celular establecida Metabolito Farmacocinética Promedicamento Ratón Toxicidad Tratamiento Tumor maligno Vía intraperitoneal Vía oral Mammalia Rodentia Vertebrata
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02R Antineoplastic agents / 002B02R02 Chemotherapy

Discipline
Pharmacological treatments
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
2305336

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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