1H-1,2,3-Triazol-1-yl thiodigalactoside derivatives as high affinity galectin-3 inhibitors
- Author
- SALAMEH, Bader A1 ; CUMPSTEY, Ian2 ; SUNDIN, Anders2 ; LEFFLER, Hakon3 ; NILSSON, Ulf J2
[1] Chemistry Department, The Hashemite University, PO Box 150459, Zarka 13115, Jordan
[2] Organic Chemistry, Lund University, PO Box 124, 221 00 Lund, Sweden
[3] Section MIG, Department of Laboratory Medicine, University of Lund, Sölvegatan 23, 223 62 Lund, Sweden - Source
Bioorganic & medicinal chemistry. 2010, Vol 18, Num 14, pp 5367-5378, 12 p
- ISSN
- 0968-0896
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Amsterdam
- Publication country
- Netherlands
- Document type
- Article
- Language
- English
- Author keyword
- Azide Galactose Galectin Inhibition Triazole
- Keyword (fr)
- Affinité Aldose Forme moléculaire Galectine Glycoprotéine Inhibition Lectine Protéine Relation structure activité Synthèse chimique Sélectivité Thioglycoside 1,2,3-Triazole-4-carboxamide dérivé
- Keyword (en)
- Affinity Aldose Molecular form Galectin Glycoprotein Inhibition Lectin Protein Structure activity relation Chemical synthesis Selectivity Thioglycoside
- Keyword (es)
- Afinidad Aldosa Forma molecular Galectina Glicoproteína Inhibición Lectina Proteína Relación estructura actividad Síntesis química Selectividad Tioglicósido
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02W Miscellaneous
- Discipline
- General pharmacology
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 23054886
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmc.2010.05.040 
https://dx.doi.org/10.1016/j.bmc.2010.05.040
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