Substituted salicylanilides as inhibitors of two-component regulatory systems in bacteria
- Author
- MACIELAG, M. J1 ; DEMERS, J. P1 ; FOLENO, B. D1 ; GOLDSCHMIDT, R. M1 ; LOELOFF, M. J1 ; WEBB, G. C1 ; BARRETT, J. F1 ; FRAGA-SPANO, S. A1 ; HLASTA, D. J1 ; JOHNSON, S. G1 ; KANOJIA, R. M1 ; RUSSELL, R. K1 ; ZHIHUA SUI1 ; WEIDNER-WELLS, M. A1 ; WERBLOOD, H1
[1] The R.W. Johnson Pharmaceutical Research Institute, 1000 Route 202, Raritan, New Jersey 08869, United States - Source
Journal of medicinal chemistry (Print). 1998, Vol 41, Num 16, pp 2939-2945 ; ref : 25 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Anilide Antibactérien Autophosphorylation Bacillus subtilis Carboxamide Chlore Composé organique Composé benzénique Enterococcus faecalis In vitro Inhibiteur enzyme Méticilline Phénols Protein kinase Relation structure activité Régulation Résistance Sporulation Staphylococcus aureus Synthèse chimique Vancomycine Benzoïque acide(2,3-dihydroxy)-3,4-dichlorophénylamide Benzoïque acide(2,3-dihydroxy)[5-chloro-4-(4-chloro-α-cyanobenzyl)-2-méthyl]phénylamide Salicylique acide dérivé Souche résistance méticilline Souche résistante vancomycine Bacillaceae Bacillales Bactérie Enzyme Micrococcaceae Micrococcales Streptococcaceae Transferases
- Keyword (en)
- Anilide Antibacterial agent Autophosphorylation Bacillus subtilis Carboxamide Chlorine Organic compounds Benzenic compound Enterococcus faecalis In vitro Enzyme inhibitor Meticillin Phenols Protein kinase Structure activity relation Regulation(control) Resistance Sporulation Staphylococcus aureus Chemical synthesis Vancomycin Bacillaceae Bacillales Bacteria Enzyme Micrococcaceae Micrococcales Streptococcaceae Transferases
- Keyword (es)
- Anilido Antibacteriano Autofosforilación Bacillus subtilis Carboxamida Cloro Compuesto orgánico Compuesto bencénico Enterococcus faecalis In vitro Inhibidor enzima Meticilina Fenoles Protein kinase Relación estructura actividad Regulación Resistencia Esporulación Staphylococcus aureus Síntesis química Vancomicina Bacillaceae Bacillales Bacteria Enzima Micrococcaceae Micrococcales Streptococcaceae Transferases
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S02 Antibacterial agents
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 2357963
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm9803572 
https://dx.doi.org/10.1021/jm9803572
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