Synthesis and in vitro anti-HIV activity of N-1,3-benzo[d]thiazol-2-yl-2-(2-oxo-2H-chromen-4-yl)acetamide derivatives using MTT method
- Author
- BHAVSAR, Dhairya1 ; TRIVEDI, Jalpa1 ; PARESH, Ladwa1 ; LODDO, Roberta2 ; SHAH, Anamik1 ; PAREKH, Shrey1 ; SAVANT, Mahesh1 ; THAKRAR, Shailesh1 ; BAVISHI, Abhay1 ; RADADIYA, Ashish1 ; VALA, Hardevsinh1 ; LUNAGARIYA, Jignesh1 ; PARMAR, Manisha1
[1] Deportment of Chemistry, Saurashtra University, Rajkot 360005, India
[2] University of Cagliari, Department of Biomedical Sciences and Technologies, Division of General Microbiology and Virology and Microbial Biotechnology, 50009042 Monserrato, Italy - Source
Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 11, pp 3443-3446, 4 p ; ref : 29 ref
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Amsterdam
- Publication country
- Netherlands
- Document type
- Article
- Language
- English
- Author keyword
- Anti-HIV activity Benzothiazole chromene derivatives MT-4 cells MTT method
- Keyword (fr)
- Activité biologique Antiviral Carboxamide Chlore Composé organique Composé nitro Dérivé de la coumarine Dérivé du benzothiazole In vitro Lactone Phénols Synthèse chimique Virus HIV1 1-Benzopyrane dérivé 1-Benzopyrane-4-acétamide(7,8-diméthyl-N-[6-nitrobenzothiazol-2-yl]-2-oxo) 1-Benzopyrane-4-acétamide(7-hydroxy-N-[6-nitrobenzothiazol-2-yl]-2-oxo) 1-Benzopyrane-4-acétamide(N-[6-chlorobenzothiazol-2-yl]-7-hydroxy-2-oxo) Acétamide dérivé Anti hiv Test MTT Lentivirus Retroviridae Virus immunodéficience humaine Virus
- Keyword (en)
- Biological activity Antiviral Carboxamide Chlorine Organic compounds Nitro compound Coumarine derivatives Benzothiazole derivatives In vitro Lactone Phenols Chemical synthesis HIV-1 virus MTT assay Lentivirus Retroviridae Human immunodeficiency virus Virus
- Keyword (es)
- Actividad biológica Antiviral Carboxamida Cloro Compuesto orgánico Compuesto nitro Benzotiazol derivado In vitro Lactona Fenoles Síntesis química HIV-1 virus Lentivirus Retroviridae Human immunodeficiency virus Virus
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S05 Antiviral agents
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 24231646
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2011.03.105 
https://dx.doi.org/10.1016/j.bmcl.2011.03.105
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