A Novel Kinase Inhibitor, INCB28060, Blocks c-MET-Dependent Signaling, Neoplastic Activities, and Cross-Talk with EGFR and HER-3
- Author
- XIANGDONG LIU1 ; QIAN WANG1 ; BOER, Jason1 ; DIAMOND, Sharon1 ; CHUNHONG HE1 ; MEIZHONG XU1 ; JINCONG ZHUO1 ; WENQING YAO1 ; NEWTON, Robert C1 ; SCHERLE, Peggy A1 ; GENGJIE YANG1 ; MARANDO, Cindy1 ; KOBLISH, Holly K1 ; HALL, Leslie M1 ; FRIDMAN, Jordan S1 ; BEHSHAD, Elham1 ; WYNN, Richard1 ; YU LI1
[1] Incyte Corporation, Wilmington, Delaware, United States - Source
Clinical cancer research (Print). 2011, Vol 17, Num 22, pp 7127-7138, 12 p ; ref : 36 ref
- CODEN
- CCREF4
- ISSN
- 1078-0432
- Scientific domain
- Medical oncology; Pharmacology drugs
- Publisher
- American Association for Cancer Research, Philadelphia, PA
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Gène onc cellulaire Inhibiteur Kinase Protooncogène Récepteur facteur croissance épiderme Transduction signal Tumeur maligne Gène met Récepteur HER3 Cancer Enzyme Transferases
- Keyword (en)
- Biological activity C-Onc gene Inhibitor Kinase Protooncogene Epidermal growth factor receptor Signal transduction Malignant tumor Human Epidermal growth factor Receptor 3 Cancer Enzyme Transferases
- Keyword (es)
- Actividad biológica Gen onc celular Inhibidor Kinase Protooncogen Receptor del factor de crecimiento epidérmico Transducción señal Tumor maligno Cáncer Enzima Transferases
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02R Antineoplastic agents
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 25229376
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1158/1078-0432.CCR-11-1157 
https://dx.doi.org/10.1158/1078-0432.CCR-11-1157
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