Coumarin-based inhibitors of HIV integrase
- Author
- ZHAO, H1 ; NEAMATI, N2 ; HONG, H1 ; MAZUMDER, A2 ; WANG, S1 ; SUNDER, S2 ; MILNE, G. W. A1 ; POMMIER, Y2 ; BURKE, T. R1
[1] Laboratory of Medicinal Chemistry, Division of Basic Sciences, National Cancer Institute, National Institutes of Health, Bethesda, Maryland 20892, United States
[2] Laboratory of Molecular Pharmacology, Division of Basic Sciences, National Cancer Institute, National Institutes of Health, Bethesda, Maryland 20892, United States - Source
Journal of medicinal chemistry (Print). 1997, Vol 40, Num 2, pp 242-249 ; ref : 17 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Antiviral Coumarine dérivé Inhibiteur enzyme Naphtalène dérivé Phénols Relation structure activité Stilbène dérivé Synthèse chimique Virus HIV1 Virus HIV2 Virus immunodéficience simienne 3,3p-Méthylènebis[1-benzopyran-2-one](α-[2-naphtyl]-4,4p,7,7p-tétrahydroxy) 3,3p-Méthylènebis[1-benzopyran-2-one](α-[stilbényl]-4,4p,7,7p-tétrahydroxy) Integrase Lentivirinae Retroviridae Virus immunodéficience humaine Virus
- Keyword (en)
- Antiviral Coumarine derivatives Enzyme inhibitor Naphthalene derivatives Phenols Structure activity relation Stilbene derivatives Chemical synthesis HIV-1 virus HIV-2 virus Simian immunodeficiency virus Lentivirinae Retroviridae Human immunodeficiency virus Virus
- Keyword (es)
- Antiviral Inhibidor enzima Naftaleno derivado Fenoles Relación estructura actividad Estilbeno derivado Síntesis química HIV-1 virus HIV-2 virus Simian immunodeficiency virus Lentivirinae Retroviridae Human immunodeficiency virus Virus
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S05 Antiviral agents
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 2541401
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm960450v 
https://dx.doi.org/10.1021/jm960450v
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