Conformational analysis of three NK1 tripeptide antagonists : A proton nuclear magnetic resonance study
- Author
- CALIENDO, G1 ; GRIECO, P1 ; PERISSUTTI, E1 ; SANTAGADA, V1 ; SAVIANO, T. G2 ; TANCREDI, T3 ; TEMUSSI, P. A2
[1] Dipartimento di Chimica Farmaceutica e Tossicologica, Università degli Studi di Napoli Federico II, via Montesano 49, 80131 Napoli, Italy
[2] Dipartimento di Chimica, Università degli Studi di Napoli Federico II, via Mezzocannone 4, 80134 Napoli, Italy
[3] Istituto Chimica MIB del CNR, Arco Felice, Napoli, Italy - Source
Journal of medicinal chemistry (Print). 1997, Vol 40, Num 4, pp 594-601 ; ref : 28 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Analyse conformationnelle Antagoniste Carboxamide Effet Overhauser Hydrogène 1 Peptide Phénylalanine Récepteur tachykinine NK1 Spectrométrie RMN Stéréoisomère D Thréonine Tripeptide Tryptophane Indole-2-carboxylique acide(octahydro) Tryptophane(1-formyl)
- Keyword (en)
- Conformational analysis Antagonist Carboxamide Overhauser effect Hydrogen 1 Peptides Phenylalanine NK1 receptor NMR spectrometry D stereoisomer Threonine Tripeptide Tryptophan
- Keyword (es)
- Análisis conformacional Antagonista Carboxamida Efecto Overhauser Péptido Fenilalanina Receptor taquikinina NK1 Espectrometría RMN Estereoisómero D Treonina Tripéptido Triptófano
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02B Neuropharmacology / 002B02B09 Neurotransmitters. Neurotransmission. Receptors / 002B02B09F Peptidergic system (neuropeptide, opioid peptide, opiates...). Adenosinergic and purinergic systems
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 2590789
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm960213s 
https://dx.doi.org/10.1021/jm960213s
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