Conformationally constrained deltorphin analogs with 2-aminotetralin-2-carboxylic acid in position 3
- Author
- TOTH, G1 ; DARULA, Z1 ; PETER, A2 ; FÜLÖP, F3 ; TOURWE, D4 ; JASPERS, H4 ; VERHEYDEN, P4 ; BÖCSKEY, Z5 ; TOTH, Z6 ; BORSODI, A1
[1] Isotope Laboratory and Institute of Biochemistry, Biological Research Center, Hungarian Academy of Sciences, P.O. Box 521, 6701 Szeged, Hungary
[2] Department of Inorganic and Analytical Chemistry, Attila József University, P.O. Box 440, 6701 Szeged, Hungary
[3] Institute of Pharmaceutical Chemistry, Albert Szent-Györgyi Medical University, P.O. Box 121, 6701 Szeged, Hungary
[4] Eenheid Organische Chemie, Vrije Universiteit Brussel, 1050 Brussels, Belgium
[5] CHINOIN Ltd., P.O. Box ll0, 1045 Budapest, Hungary
[6] Alkaloida Chemical Factory Ltd., P.O. Box 1, 4440 Tiszavasvári, Hungary - Source
Journal of medicinal chemistry (Print). 1997, Vol 40, Num 6, pp 990-995 ; ref : 39 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Affinité Animal Conformation Heptapeptide In vitro Naphtalène dérivé Naphtalène(1,2,3,4-tétrahydro) Peptide Phase solide Relation structure activité Récepteur opiacé δ Synthèse chimique Synthèse peptidique Glycine(tyrosyl-D-alanyl-[2-amino-1,2,3,4-tétrahydro-2-naphtoyl]-glutamyl-isoleucyl-isoleucyl) amide
- Keyword (en)
- Affinity Animal Conformation Heptapeptide In vitro Naphthalene derivatives Naphthalene(1,2,3,4-tetrahydro) Peptides Solid phase Structure activity relation Opiate receptor δ Chemical synthesis Peptide synthesis
- Keyword (es)
- Afinidad Animal Conformación Heptapéptido In vitro Naftaleno derivado Naftaleno(1,2,3,4-tetrahidro) Péptido Fase sólida Relación estructura actividad Receptor opiáceo δ Síntesis química Síntesis peptídica
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02B Neuropharmacology / 002B02B09 Neurotransmitters. Neurotransmission. Receptors / 002B02B09F Peptidergic system (neuropeptide, opioid peptide, opiates...). Adenosinergic and purinergic systems
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 2602401
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm9602726 
https://dx.doi.org/10.1021/jm9602726
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