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The activity of GR205171, a potent non-peptide tachykinin NK1 receptor antagonist, in the trigeminovascular system

Author
POLLEY, J. S1 ; GASKIN, P. J1 ; PERREN, M. J1 ; CONNOR, H. E2 ; WARD, P3 ; BEATTIE, D. T1
[1] Systems Biology, Glaxo Wellcome Medicines Research Centre, Gunnels Woods Road, Stevenage, Herts SG1 2NY, United Kingdom
[2] Receptor Pharmacology, Glaxo Wellcome Medicines Research Centre, Gunnels Woods Road, Stevenage, Herts, SG1 2NY, United Kingdom
[3] Medicinal chemistry, Glaxo Wellcome Medicines Research Centre, Gunnels Wood Road, Stevenage, Herts SG1 2NY, United Kingdom
Source

Regulatory peptides. 1997, Vol 68, Num 1, pp 23-29 ; ref : 25 ref

CODEN
REPPDY
ISSN
0167-0115
Scientific domain
Endocrinology; Gastroenterology; Neurology
Publisher
Elsevier, Amsterdam / Elsevier, Shannon
Publication country
Netherlands
Document type
Article
Language
English
Keyword (fr)
Animal Antagoniste Chimiothérapie Douleur Extravasation Migraine Noyau trijumeau Récepteur tachykinine NK1 Tachykinine Traitement GR205171 Appareil circulatoire pathologie Cérébrovasculaire pathologie Encéphale pathologie Encéphale Système nerveux central pathologie Système nerveux central Système nerveux pathologie Vaisseau sanguin pathologie
Keyword (en)
Animal Antagonist Chemotherapy Pain Extravasation Migraine Trigeminal nucleus NK1 receptor Tachykinin Treatment Cardiovascular disease Cerebrovascular disease Cerebral disorder Brain (vertebrata) Central nervous system disease Central nervous system Nervous system diseases Vascular disease
Keyword (es)
Animal Antagonista Quimioterapia Dolor Extravasación Jaqueca Núcleo trigeminal Receptor taquikinina NK1 Taquikinina Tratamiento Aparato circulatorio patología Vaso sanguíneo encéfalo patología Encéfalo patología Encéfalo Sistema nervosio central patología Sistema nervioso central Sistema nervioso patología Vaso sanguíneo patología
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02F Cardiovascular system / 002B02F04 Vasodilator agents. Cerebral vasodilators

Discipline
Pharmacological treatments
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
2602626

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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