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Optimizing solubility: Kinetic versus thermodynamic solubility temptations and risks

Author
SAAL, Christoph1 ; CHRISTINE PETEREIT, Anna1
[1] Merck KGaA, Frankfurter Strasse 250, 64293 Darmstadt, Germany
Source

European journal of pharmaceutical sciences. 2012, Vol 47, Num 3, pp 589-595, 7 p ; ref : 1/4 p

ISSN
0928-0987
Scientific domain
Pharmacology drugs
Publisher
Elsevier, Kindlington
Publication country
United Kingdom
Document type
Article
Language
English
Author keyword
Crystallinity Dissolution Precipitation Solid state Solubility Thermodynamics
Keyword (fr)
Cinétique Cristallinité Dissolution Etat solide Etude comparative Facteur risque Précipitation Solubilité Technologie pharmaceutique Thermodynamique Propriété physicochimique
Keyword (en)
Kinetics Crystallinity Dissolution Solid state Comparative study Risk factor Precipitation Solubility Pharmaceutical technology Thermodynamics Physicochemical properties
Keyword (es)
Cinética Cristalinidad Disolución Estado sólido Estudio comparativo Factor riesgo Precipitación Solubilidad Tecnología farmacéutica Termodinámica Propiedad fisicoquímica
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02A General pharmacology / 002B02A03 Pharmaceutical technology. Pharmaceutical industry

Discipline
General pharmacology
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
26429201

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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