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The novel oral imatinib microemulsions: physical properties, cytotoxicity activities and improved Caco-2 cell permeability

Author
GUNDOGDU, Evren1 ; KARASULU, Hatice Yesim2 ; KOKSAL, Cinel3 4 ; KARASULU, Ercüment1 3
[1] Department of Biopharmaceutics and Pharmacokinetics, Faculty of Pharmacy, Ege University, Izmir 35100, Turkey
[2] Department of Pharmaceutical Technology, Faculty of Pharmacy, Ege University, Izmir 35100, Turkey
[3] Center for Drug Research & Development and Pharmacokinetic Applications, Ege University, Izmir 35100, Turkey
[4] Department of Biology, Faculty of Science, Ege University, Bornova, Izmir 35100, Turkey
Source

Journal of microencapsulation. 2013, Vol 30, Num 2, pp 132-142, 11 p ; ref : 3/4 p

CODEN
JOMIEF
ISSN
0265-2048
Scientific domain
Nanotechnologies, nanostructures, nanoobjects; Pharmacology drugs
Publisher
Informa, Colchester
Publication country
United Kingdom
Document type
Article
Language
English
Author keyword
cell culture imatinib microemulsion permeability
Keyword (fr)
Anticancéreux Culture cellulaire Cytotoxicité Exercice physique Imatinib In vitro Intestin Microémulsion Perméabilité Propriété physique Technologie pharmaceutique Voie orale Enzyme Inhibiteur de la tyrosine kinase Inhibiteur enzyme Protein-tyrosine kinase Transferases
Keyword (en)
Antineoplastic agent Cell culture Cytotoxicity Physical exercise Imatinib In vitro Gut Microemulsion Permeability Physical properties Pharmaceutical technology Oral administration Enzyme Tyrosine kinase inhibitor Enzyme inhibitor Protein-tyrosine kinase Transferases
Keyword (es)
Anticanceroso Cultivo celular Citotoxicidad Ejercicio físico Imatinib In vitro Intestino Microemulsión Permeabilidad Propiedad física Tecnología farmacéutica Vía oral Enzima Inhibidor tyrosine kinase Inhibidor enzima Protein-tyrosine kinase Transferases
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02A General pharmacology / 002B02A03 Pharmaceutical technology. Pharmaceutical industry

Discipline
General pharmacology
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
27811384

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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