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Cross-resistance to antifolates in multidrug resistant cell lines with P-glycoprotein or multidrug resistance protein expression

Author
VAN TRIEST, B1 ; PINEDO, H. M1 ; TELLEMAN, F1 ; VAN DER WILT, C. L1 ; JANSEN, G1 ; PETERS, G. J1
[1] Department of Medical Oncology, University Hospital Vrije Universiteit, PO Box 7057, 1007 MB Amsterdam, Netherlands
Source

Biochemical pharmacology. 1997, Vol 53, Num 12, pp 1855-1866 ; ref : 63 ref

CODEN
BCPCA6
ISSN
0006-2952
Scientific domain
Biochemistry, molecular biology, biophysics; Pharmacology drugs; Physiology, morphology
Publisher
Elsevier Science, New York, NY
Publication country
United States
Document type
Article
Language
English
Keyword (fr)
Anthracyclines Anticancéreux Antifolate Bronchopulmonaire Carcinome Cellule tumorale Doxorubicine Fluoropyrimidine dérivé Fluorouracil Glycoprotéine P Homme In vitro Inhibiteur enzyme Lignée cellulaire établie Résistance croisée Résistance multiple Thymidylate synthase Transport biologique Transport membranaire Lignée SW1573 Appareil respiratoire pathologie Bronche pathologie Enzyme Methyltransferases Poumon pathologie Transferases Tumeur maligne
Keyword (en)
Anthracyclins Antineoplastic agent Antifolate Bronchopulmonary Carcinoma Tumor cell Doxorubicin Fluoropyrimidine derivatives Fluorouracil P Glycoprotein Human In vitro Enzyme inhibitor Established cell line Cross resistance Multiple resistance Thymidylate synthase Biological transport Membrane transport Respiratory disease Bronchus disease Enzyme Methyltransferases Lung disease Transferases Malignant tumor
Keyword (es)
Antraciclinas Anticanceroso Antifolato Broncopulmonar Carcinoma Célula tumoral Doxorubicina Fluoropirimidina derivado Fluorouracilo Glycoproteina P Hombre In vitro Inhibidor enzima Línea celular establecida Resistencia cruzada Resistencia múltiple Thymidylate synthase Transporte biológico Transporte membranal Aparato respiratorio patología Bronquio patología Enzima Methyltransferases Pulmón patología Transferases Tumor maligno
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02R Antineoplastic agents / 002B02R01 General aspects

Discipline
Pharmacological treatments
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
2781832

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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