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Potential irreversible ligands for opioid receptors. Cinnamoyl derivatives of β-naltrexamine

Author
DERRICK, I1 ; LEWIS, J. W1 ; MOYNIHAN, H. A1 ; BROADBEAR, J; WOODS, J. H
[1] School of Chemistry, University of Bristol, Bristol BS8 1TS, United Kingdom
Source

Journal of pharmacy and pharmacology. 1996, Vol 48, Num 2, pp 192-196 ; ref : 19 ref

CODEN
JPPMAB
ISSN
0022-3573
Scientific domain
Pharmacology drugs
Publisher
Pharmaceutical Press, Wallingford
Publication country
United Kingdom
Document type
Article
Language
English
Keyword (fr)
Animal Antagoniste Appareil digestif Appareil urogénital Canal déférent Cobaye Fixation biologique Iléon In vitro In vivo Intestin Irréversible Nociception Récepteur opiacé Souris BU 42 BU 59 BU 60 Naltrexamine dérivé Mammalia Rodentia Vertebrata
Keyword (en)
Animal Antagonist Digestive system Urogenital system Vas deferens Guinea pig Biological fixation Ileum In vitro In vivo Gut Irreversible Nociception Opiate receptor Mouse Mammalia Rodentia Vertebrata
Keyword (es)
Animal Antagonista Aparato digestivo Aparato urogenital Canal deferente Cobayo Fijación biológica Ileon In vitro In vivo Intestino Irreversible Nocicepción Receptor opiáceo Ratón Mammalia Rodentia Vertebrata
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02B Neuropharmacology / 002B02B09 Neurotransmitters. Neurotransmission. Receptors / 002B02B09F Peptidergic system (neuropeptide, opioid peptide, opiates...). Adenosinergic and purinergic systems

Discipline
Pharmacological treatments
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
3033014

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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