Iterative protein structure-based drug design and synthesis of HIV protease inhibitors
- Author
- KALISH, V1 ; KALDOR, S; MUSICK, L1 ; BOR-WEN WU1 ; KEN SU; SHETTY, B1 ; TATLOCK, J1 ; DAVIES, J1 ; HAMMOND, M; DRESSMAN, B; FRITZ, J; APPELT, K1 ; REICH, S1
[1] Agouron Pharmaceuticals, San Diego CA 92121, United States - Conference title
- International symposium on medicinal chemistry
- Conference name
- International symposium on medicinal chemistry (13 ; Paris 1994)
- Author (monograph)
- MULLER, Jean-Claude (Editor)
European Federation for Medicinal Chemistry, Europe (Funder/Sponsor)
American Chemical Society, Washington DC, United States (Funder/Sponsor)
International Union of Pure and Applied Chemistry, International (Funder/Sponsor) - Source
European journal of medicinal chemistry. 1995, Vol 30, pp 201s-214s ; SUP ; ref : 18 ref
- CODEN
- EJMCA5
- ISSN
- 0223-5234
- Scientific domain
- Organic chemistry; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Conference Paper
- Language
- English
- Keyword (fr)
- Animal Antiviral Biodisponibilité Hydroxysulfure organique Inhibiteur enzyme Isoquinoléine dérivé Modèle moléculaire Modélisation Phénols Proteinases Relation structure activité Structure cristalline Virus immunodéficience humaine Voie orale AG 1343 Benzoïque acide dérivé LY 289612 Enzyme Hydrolases Lentivirinae Retroviridae Virus
- Keyword (en)
- Animal Antiviral Bioavailability Organic hydroxysulfide Enzyme inhibitor Isoquinoline derivatives Molecular model Modeling Phenols Proteinases Structure activity relation Crystalline structure Human immunodeficiency virus Oral administration Enzyme Hydrolases Lentivirinae Retroviridae Virus
- Keyword (es)
- Animal Antiviral Biodisponibilidad Hidroxisulfuro orgánico Inhibidor enzima Isoquinoleína Modelo molecular Modelización Fenoles Proteinases Relación estructura actividad Estructura cristalina Human immunodeficiency virus Vía oral Enzima Hydrolases Lentivirinae Retroviridae Virus
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S05 Antiviral agents
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 3567530
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/S0223-5234(23)00125-3 
https://dx.doi.org/10.1016/S0223-5234(23)00125-3
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