Structure and conformation of the muscarinic agonists 3-(3-amino-1,2,4-oxadiazol-5-yl)-1-azabicyclo[2.2.2]octane and 1,2,5,6-tetrahydro-1-methyl-3-pyridinecarbox-aldehyde oxime and related tertiary amine, quaternary ammonium and sulfonium analogues
- Author
- KOOIJMAN, H1 ; KANTERS, J. A1 ; KROON, J1 ; KELDER, J
[1] Rijksuniv. Utrecht, Vakgroep Kristal Structuurchemie, 3584 CH Utrecht, Netherlands - Source
Acta crystallographica. Section B, Structural science. 1993, Vol 49, Num 2, pp 356-366 ; ref : 43 ref
- CODEN
- ASBSDK
- ISSN
- 0108-7681
- Scientific domain
- Crystallography
- Publisher
- Blackwell, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Keyword (fr)
- Agoniste Ammonium quaternaire composé Cation organique Composé bicyclique Conformation Cycle 5 chaînons Cycle 6 chaînons Etude comparative Etude expérimentale Guanidines Hétérocycle azote angulaire Hétérocycle azote Hétérocycle oxygène azote Oxime Relation structure activité Récepteur muscarinique Structure cristalline Structure moléculaire XRD L-660863 Org 31956 Pyridine-«3»-carbaldéhyde(«1»-méthyl-«1,2,5,6»-tétrahydro) oxime «1»-Azabicyclo[«2.2.2»]octane dérivé Composé organique
- Keyword (en)
- Agonist Quaternary ammonium compound Organic cation Bicyclic compound Conformation Five membered ring Six membered ring Comparative study Experimental study Guanidines Angular nitrogen heterocycle Nitrogen heterocycle Oxygen nitrogen heterocycle Oximes Structure-activity relationships Muscarinic receptor Crystal structure Molecular structure XRD Organic compounds
- Keyword (es)
- Agonista Amonio cuaternario compuesto Catión orgánico Compuesto bicíclico Conformación Ciclo 5 eslabones Ciclo 6 eslabones Estudio comparativo Heterociclo nitrógeno angular Heterociclo nitrógeno Heterociclo oxígeno nitrógeno Receptor muscarínico
- Classification
- Pascal
- 001 Exact sciences and technology / 001B Physics / 001B60 Condensed matter: structure, mechanical and thermal properties / 001B60A Structure of solids and liquids; crystallography / 001B60A10 X-ray diffraction and scattering / 001B60A10N Single-crystal and powder diffraction
- Pascal
- 001 Exact sciences and technology / 001B Physics / 001B60 Condensed matter: structure, mechanical and thermal properties / 001B60A Structure of solids and liquids; crystallography / 001B60A66 Structure of specific crystalline solids / 001B60A66H Organic compounds / 001B60A66H3 Heterocyclic compounds
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02B Neuropharmacology / 002B02B09 Neurotransmitters. Neurotransmission. Receptors / 002B02B09B Cholinergic system
- Discipline
- Pharmacological treatments Physics of condensed state : structure, mechanical and thermal properties
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 3755168
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1107/S0108768192008383 
https://dx.doi.org/10.1107/S0108768192008383
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