Synthesis and anticonvulsant activities of α-heterocyclic α-acetamido-N-benzylacetamide derivatives
- Author
- KOHN, H1 ; SAWHNEY, K. N1 ; BARDEL, P1 ; ROBERTSON, D. W; LEANDER, J. D
[1] Univ. Houston, dep. chemistry, Houston TX 77204-5641, United States - Source
Journal of medicinal chemistry (Print). 1993, Vol 36, Num 22, pp 3350-3360 ; ref : 29 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Aminoamide Animal Anticonvulsivant Cycle 5 chaînons Hétérocycle oxygène azote Hétérocycle oxygène Hétérocycle soufre azote Relation structure activité Souris Substitution nucléophile Furane-2-acétique acide(α-acétamido) benzylamide Oxazole-2-acétique acide(α-acétamido) benzylamide Thiazole-2-acétique acide(α-acétamido) benzylamide Mammalia Rodentia Vertebrata
- Keyword (en)
- Aminoamide Animal Anticonvulsant Five membered ring Oxygen nitrogen heterocycle Oxygen heterocycle Sulfur nitrogen heterocycle Structure activity relation Mouse Nucleophilic substitution Mammalia Rodentia Vertebrata
- Keyword (es)
- Aminoamida Animal Anticonvulsivante Ciclo 5 eslabones Heterociclo oxígeno nitrógeno Heterociclo oxígeno Heterociclo azufre nitrógeno Relación estructura actividad Ratón Substitución nucleófila Mammalia Rodentia Vertebrata
- Classification
- Pascal
- 001 Exact sciences and technology / 001C Chemistry / 001C03 Organic chemistry / 001C03C Preparations and properties / 001C03C06 Heterocyclic compounds / 001C03C06D Heterocyclic compounds with n hetero atom and also o and/or s, se, te hetero atoms
- Discipline
- Organic chemistry
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 3809967
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm00074a016 
https://dx.doi.org/10.1021/jm00074a016
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