Synthesis and antibacterial activity of thiazolopyrazine-incorporated tetracyclic quinolone antibacterials
- Author
- INOUE, Y; KONDO, H; TAGUCHI, M; JINBO, Y; SAKAMOTO, F; TSUKAMOTO, G
Kanebo Ltd, New Drug Research Laboratories, Miyakojima-ku, Osaka 534, Japan - Source
Journal of medicinal chemistry (Print). 1994, Vol 37, Num 5, pp 586-592 ; ref : 12 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Amine secondaire Antibactérien Composé aromatique Composé tétracyclique Cétoacide Hétérocycle soufre azote In vitro In vivo Pipérazine dérivé Souris 1-Thia-4,9b-diazacyclopenta[cd]phénalène-9-carboxylique acide(5-dialkylamino-3,4-dihydro-6-fluoro-4-méthyl-8-oxo) Acétone(1,3-dichloro) Ammonium(triéthyl) dithiocarbamate(N-[2,3,4-trifluorophényl]) Thiazolo[3,4-a]quinoxaline dérivé Fluor Composé organique Mammalia Rodentia Vertebrata
- Keyword (en)
- Biological activity Secondary amine Antibacterial agent Aromatic compound Tetracyclic compound Ketoacid Sulfur nitrogen heterocycle In vitro In vivo Piperazine derivatives Mouse Fluorine Organic compounds Mammalia Rodentia Vertebrata
- Keyword (es)
- Actividad biológica Amina secundaria Antibacteriano Compuesto aromático Compuesto tetracíclico Cetoácido Heterociclo azufre nitrógeno In vitro In vivo Ratón Fluor Compuesto orgánico Mammalia Rodentia Vertebrata
- Classification
- Pascal
- 001 Exact sciences and technology / 001C Chemistry / 001C03 Organic chemistry / 001C03C Preparations and properties / 001C03C06 Heterocyclic compounds / 001C03C06D Heterocyclic compounds with n hetero atom and also o and/or s, se, te hetero atoms
- Discipline
- Organic chemistry
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 3968026
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm00031a007 
https://dx.doi.org/10.1021/jm00031a007
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