Synthesis of naltrexone-derived δ-opioid antagonists. Role of conformation of the δ adress moiety
- Author
- PORTOGHESE, P. S; SULTANA, M; MOE, S. T; TAKEMORI, A. E
Univ. Minnesota, coll. pharmacy, dep. medicinal, Minneapolis MN 55455, United States - Source
Journal of medicinal chemistry (Print). 1994, Vol 37, Num 5, pp 579-585 ; ref : 31 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Analogue Animal Antagoniste analgésique narcotique Antagoniste Benzène Composé aromatique Conformation Fixation biologique In vitro In vivo Indole dérivé Muscle lisse Naltrexone Récepteur opiacé δ Synthèse chimique
- Keyword (en)
- Biological activity Analog Animal Narcotic antagonist Antagonist Benzene Aromatic compound Conformation Biological fixation In vitro In vivo Indole derivatives Smooth muscle Opiate receptor δ Chemical synthesis
- Keyword (es)
- Actividad biológica Análogo Animal Antagonista narcótico Antagonista Benceno Compuesto aromático Conformación Fijación biológica In vitro In vivo Indol derivado Músculo liso Receptor opiáceo δ Síntesis química
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02B Neuropharmacology / 002B02B09 Neurotransmitters. Neurotransmission. Receptors / 002B02B09F Peptidergic system (neuropeptide, opioid peptide, opiates...). Adenosinergic and purinergic systems
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 3980192
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm00031a006 
https://dx.doi.org/10.1021/jm00031a006
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