Synthesis and biological evaluation of 2',3'-dideoxy-L-pyrimidine nucleosides as potential antiviral agents against human immunodeficiency virus (HIV) and hepatitis B virus (HBV)
- Author
- TAI-SHUN LIN; MEI-ZHEN LUO; MAO-CHIN LIU; BALAKRISHNA PAI, S; DUTSCHMAN, G. E; YUNG-CHI CHENG
Yale univ. school medicine, comprehensive cancer cent., dep. pharmacology, New Haven CT 06510, United States - Source
Journal of medicinal chemistry (Print). 1994, Vol 37, Num 6, pp 798-803 ; ref : 36 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Anomère Antiviral Didésoxynucléoside In vitro Pyrimidine nucléoside Stéréoisomère L Virus HIV1 Virus hépatite B Cytosine(1-[2,3-didésoxy-β-L-glycéro-pentofuranosyl]) Cytosine(1-[2,3-didésoxy-β-L-glycéro-pentofuranosyl]-5-fluoro) Hepadnaviridae Lentivirinae Retroviridae Virus immunodéficience humaine Virus
- Keyword (en)
- Biological activity Anomer Antiviral Dideoxynucleoside In vitro Pyrimidine nucleoside L stereoisomer HIV-1 virus Hepatitis B virus Hepadnaviridae Lentivirinae Retroviridae Human immunodeficiency virus Virus
- Keyword (es)
- Actividad biológica Anómero Antiviral Didesoxinucleósido In vitro Pirimidina nucleósido Estereoisómero L HIV-1 virus Hepatitis B virus Hepadnaviridae Lentivirinae Retroviridae Human immunodeficiency virus Virus
- Classification
- Pascal
- 001 Exact sciences and technology / 001C Chemistry / 001C03 Organic chemistry / 001C03C Preparations and properties / 001C03C07 Carbohydrates. Nucleosides and nucleotides / 001C03C07B Nucleosides, nucleotides and oligonucleotides
- Discipline
- Organic chemistry
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 4005298
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm00032a013 
https://dx.doi.org/10.1021/jm00032a013
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