Synthesis and anticholinergic activity of the four stereoisomers of 4-(dimethylamino)-2-phenyl-2-(2-pyridyl)pentanamide
- Author
- OYASU, H; NAGANO, M; AKAHANE, A; TOMOI, M; TADA, T; MATSUO, M
Fujisawa Pharmaceutical Co. Ltd, New Drug Research Laboratories, R & D div., Yodogawa-ku, Osaka 532, Japan - Source
Journal of medicinal chemistry (Print). 1994, Vol 37, Num 9, pp 1378-1381 ; ref : 19 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Aminoamide Composé aliphatique Composé organique Configuration absolue Diastéréoisomère Diffraction RX Dédoublement optique Etude expérimentale In vitro Parasympatholytique Pyridine dérivé Structure cristalline Structure moléculaire Stéréoisomère Valérique acide(4-diméthylamino-2-phényl-2-[2-pyridyl]) amide bornane-10-sulfonate(2-oxo) Valérique acide(4-diméthylamino-2-phényl-2-[2-pyridyl]) amide succinate(dibenzoyloxy) Valérique acide(4-diméthylamino-2-phényl-2-[2-pyridyl]) amide
- Keyword (en)
- Biological activity Aminoamide Aliphatic compound Organic compounds Absolute configuration Diastereomer X ray diffraction Optical resolution Experimental study In vitro Parasympatholytic Pyridine derivatives Crystalline structure Molecular structure Stereoisomer
- Keyword (es)
- Actividad biológica Aminoamida Compuesto alifático Compuesto orgánico Configuración absoluta Diasteréomero Difracción RX Desdoblamiento óptico Estudio experimental In vitro Parasimpatolítico Piridina derivado Estructura cristalina Estructura molecular Estereoisómero
- Classification
- Pascal
- 001 Exact sciences and technology / 001B Physics / 001B60 Condensed matter: structure, mechanical and thermal properties / 001B60A Structure of solids and liquids; crystallography / 001B60A66 Structure of specific crystalline solids / 001B60A66H Organic compounds / 001B60A66H3 Heterocyclic compounds
- Pascal
- 001 Exact sciences and technology / 001C Chemistry / 001C03 Organic chemistry / 001C03C Preparations and properties / 001C03C06 Heterocyclic compounds / 001C03C06B Heterocyclic compounds with only one n hetero atom and condensed derivatives
- Discipline
- Organic chemistry Physics of condensed state : structure, mechanical and thermal properties
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 4066067
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm00035a019 
https://dx.doi.org/10.1021/jm00035a019
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