Oxadiazoles as bioisosteric transformations of carboxylic functionalities. I
- Author
- ANDERSEN, K. E; JØRGENSEN, A. S; BRÆSTRUP, C
Novo Nordisk A/S, CNS div., 2760 Maaloev, Denmark - Source
European journal of medicinal chemistry. 1994, Vol 29, Num 5, pp 393-399 ; ref : 11 ref
- CODEN
- EJMCA5
- ISSN
- 0223-5234
- Scientific domain
- Organic chemistry; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Composé bicyclique Hétérocycle azote angulaire Hétérocycle oxygène azote In vivo Oxadiazole dérivé Récepteur benzodiazépinique Souris Pyrazolo[1,5-a]pyrimidine(3-[3-méthyl-1,2,4-oxadiazol-5-yl]-7-[3-(trifluorométhyl)phényl]) Pyrrolo[1,2-a]pyrimidine-8-carbonitrile(6,7-diméthyl-4-[3-(trifluorométhyl)phényl]) Fluor Composé organique Mammalia Rodentia Vertebrata
- Keyword (en)
- Biological activity Bicyclic compound Angular nitrogen heterocycle Oxygen nitrogen heterocycle In vivo Oxadiazole derivatives Benzodiazepine receptor Mouse Fluorine Organic compounds Mammalia Rodentia Vertebrata
- Keyword (es)
- Actividad biológica Compuesto bicíclico Heterociclo nitrógeno angular Heterociclo oxígeno nitrógeno In vivo Oxadiazol derivado Receptor benzodiazepínico Ratón Fluor Compuesto orgánico Mammalia Rodentia Vertebrata
- Classification
- Pascal
- 001 Exact sciences and technology / 001C Chemistry / 001C03 Organic chemistry / 001C03C Preparations and properties / 001C03C06 Heterocyclic compounds / 001C03C06C Heterocyclic compounds with several n hetero atoms in the same ring, in separated rings or in fused rings
- Discipline
- Organic chemistry
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 4149139
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/0223-5234(94)90065-5 
https://dx.doi.org/10.1016/0223-5234(94)90065-5
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