Synthesis and characterization of selective fluorescent ligands for the neurokinin NK2 receptor
- Author
- BRADSHAW, C. G; CESZKOWSKI, K; TURCATTI, G; BERESFORD, I. J. M; CHOLLET, A
Glaxo inst. molecular biology, 1228 Plan-les-Ouates, France - Source
Journal of medicinal chemistry (Print). 1994, Vol 37, Num 13, pp 1991-1995 ; ref : 20 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Composé bicyclique Composé fluorescent Composé nitro Heptapeptide Hétérocycle oxygène azote Modélisation Phase solide Récepteur tachykinine NK2 Synthèse peptidique 2,1,3-Benzooxadiazole dérivé Norleucine([2-benzamido-4-(7-nitro-2,1,3-benzooxadiazol-4-ylamino)butyryl]-alanyl-D-tryptophyl-phénylalanyl-D-prolyl-prolyl) amide Norleucine([Nα-benzoyl-Nδ-(7-nitro-2,1,3-benzooxadiazol-4-yl)lysyl]-alanyl-D-tryptophyl-phénylalanyl-D-prolyl-prolyl) amide Norleucine([Nα-benzoyl-Nε-(7-nitro-2,1,3-benzooxadiazol-4-yl)ornithyl]-alanyl-D-tryptophyl-phénylalanyl-D-prolyl-prolyl) amide
- Keyword (en)
- Biological activity Bicyclic compound Fluorescent compound Nitro compound Heptapeptide Oxygen nitrogen heterocycle Modeling Solid phase NK2 receptor Peptide synthesis
- Keyword (es)
- Actividad biológica Compuesto bicíclico Compuesto fluorescente Compuesto nitro Heptapéptido Heterociclo oxígeno nitrógeno Modelización Fase sólida Receptor taquikinina NK2 Síntesis peptídica
- Classification
- Pascal
- 001 Exact sciences and technology / 001C Chemistry / 001C03 Organic chemistry / 001C03C Preparations and properties / 001C03C08 Peptides
- Discipline
- Organic chemistry
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 4160225
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm00039a012 
https://dx.doi.org/10.1021/jm00039a012
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