Substituted 1,3-dipropylxanthines as irreversible antagonists of A1 adenosine receptors
- Author
- SCAMMELS, P. J1 ; BAKER, S. P; BELARDINELLI, L; OLSSON, R. A1
[1] Univ. South Florida, dep. internal medicine, Tampa FL 33612, United States - Source
Journal of medicinal chemistry (Print). 1994, Vol 37, Num 17, pp 2704-2712 ; ref : 37 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Antagoniste Carboxamide Composé benzénique Composé bicyclique Ester Halogénure sulfonyle Hétérocycle azote Purine dérivé Récepteur adénosinique A1 Xanthine dérivé Xanthine(1,3-dipropyl-8-[4-(fluorosulfonyl)benzamidométhyl]) Xanthine(8-cyclopentyl-3-[3-(4-[fluorosulfonyl]benzoyloxy)propyl])
- Keyword (en)
- Biological activity Antagonist Carboxamide Benzenic compound Bicyclic compound Ester Sulfonyl halide Nitrogen heterocycle Purine derivatives A1 Adenosine receptor Xanthine derivatives
- Keyword (es)
- Actividad biológica Antagonista Carboxamida Compuesto bencénico Compuesto bicíclico Ester Halogenuro sulfonilo Heterociclo nitrógeno Purina derivado Receptor adenosínico A1 Xantina derivado
- Classification
- Pascal
- 001 Exact sciences and technology / 001C Chemistry / 001C03 Organic chemistry / 001C03C Preparations and properties / 001C03C06 Heterocyclic compounds / 001C03C06C Heterocyclic compounds with several n hetero atoms in the same ring, in separated rings or in fused rings
- Discipline
- Organic chemistry
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 4179432
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm00043a010 
https://dx.doi.org/10.1021/jm00043a010
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