Synthesis of androst-5-en-7-ones and androsta-3,5-dien-7-ones and their related 7-deoxy analogs as conformational and catalytic probes for the active site of aromatase
- Author
- NUMAZAWA, M; MUTSUMI, A; TACHIBANA, M; HOSHI, K
Tohoku coll. pharmacy, Aobaku, Sendai 981, Japan - Source
Journal of medicinal chemistry (Print). 1994, Vol 37, Num 14, pp 2198-2205 ; ref : 33 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Anticancéreux Enone Estrogen synthase Homme Hormone stéroïde In vitro Inhibiteur enzyme Inhibition compétitive Placenta Relation structure activité Synthèse chimique Androst-5-én-7-one Androsta-3,5-dién-7-one Enzyme
- Keyword (en)
- Antineoplastic agent Enone Estrogen synthase Human Steroid hormone In vitro Enzyme inhibitor Competitive inhibition Placenta Structure activity relation Chemical synthesis Enzyme
- Keyword (es)
- Anticanceroso Enona Estrogen synthase Hombre Hormona esteroide In vitro Inhibidor enzima Inhibición competitiva Placenta Relación estructura actividad Síntesis química Enzima
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02R Antineoplastic agents / 002B02R01 General aspects
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 4191153
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm00040a012 
https://dx.doi.org/10.1021/jm00040a012
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