Synthesis and opioid activity of 7-oxygenated 2,3,4,4a,5,6,7,7a-octahyro-1H-benzofuro[3,2-e]isoquinolin-9-ols
- Author
- CHEN-YU CHENG; LING-WEI HSIN; MING-CHENG TSAI; SCHMIDT, W. K; SMITH, C; TAM, S. W
National Taiwan univ., coll. medicine, school pharmacy, Taipei 10018, Taiwan, Province of China - Source
Journal of medicinal chemistry (Print). 1994, Vol 37, Num 19, pp 3121-3127 ; ref : 22 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Analgésique Composé aromatique Composé tétracyclique Hétérocycle oxygène azote In vivo Récepteur opiacé Récepteur sigma Souris Benzo[3,2-e]isoquinoléin-7-one(3-cyclopropyl-9-hydroxy-octahydro) Benzo[3,2-e]isoquinoléine-7α,9-diol(3-cyclopropyl-octahydro) Pyridinium(1-cyclopropylméthyl-3-[2-(éthoxycarbonyl)éthyl]-4-[2-(éthoxycarbonylméthoxy)-3-méthoxyphényl]) bromure Mammalia Rodentia Vertebrata
- Keyword (en)
- Biological activity Analgesic Aromatic compound Tetracyclic compound Oxygen nitrogen heterocycle In vivo Opiate receptor Sigma receptor Mouse Mammalia Rodentia Vertebrata
- Keyword (es)
- Actividad biológica Analgésico Compuesto aromático Compuesto tetracíclico Heterociclo oxígeno nitrógeno In vivo Receptor opiáceo Receptor sigma Ratón Mammalia Rodentia Vertebrata
- Classification
- Pascal
- 001 Exact sciences and technology / 001C Chemistry / 001C03 Organic chemistry / 001C03C Preparations and properties / 001C03C06 Heterocyclic compounds / 001C03C06D Heterocyclic compounds with n hetero atom and also o and/or s, se, te hetero atoms
- Discipline
- Organic chemistry
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 4231293
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm00045a017 
https://dx.doi.org/10.1021/jm00045a017
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