Synthesis and antimicrobial activity of DNA-gyrase inhibiting derivatives of 4-oxo-1,4-dihydro-3-pyridinecarboxylic acid
- Author
- BASSINI, C; BISMARA, C; XERRI, L; CARLESSO, R; FERIANI, A; GAVIRAGHI, G; MARCHIORO, C; PERBONI, A; SHAW, R. E; TAMBURINI, B; TARZIA, G
GLAXO S.p.a. Research Laboratories, dep. chemistry, 37100 Verona, Italy - Conference name
- Meeting on heterocyclic structures in medicinal chemistry research (5 ; Palermo 1992-05-17)
- Source
Il Farmaco (Pavia). 1993, Vol 48, Num 2, pp 159-189 ; ref : 53 ref
- ISSN
- 0014-827X
- Scientific domain
- Pharmacology drugs
- Publisher
- Elsevier Science, Lausanne
- Publication country
- Switzerland
- Document type
- Conference Paper
- Language
- English
- Keyword (fr)
- Analogue Antibactérien Bactérie Gram positif DNA topoisomerase (ATP-hydrolysing) In vitro Inhibiteur enzyme Relation structure activité Synthèse chimique Test sensibilité médicamenteuse Nicotinique acide(1,4-dihydro-4-oxo) Quinolone dérivé Enzyme
- Keyword (en)
- Analog Antibacterial agent Gram positive bacteria DNA topoisomerase (ATP-hydrolysing) In vitro Enzyme inhibitor Structure activity relation Chemical synthesis Drug susceptibility test Quinolone derivative Enzyme
- Keyword (es)
- Análogo Antibacteriano Bacteria Gram positiva DNA topoisomerase (ATP-hydrolysing) In vitro Inhibidor enzima Relación estructura actividad Síntesis química Prueba sensibilidad medicamentosa Enzima
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S02 Antibacterial agents
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 4926229
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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