An efficient synthesis of hydroxyethylene dipeptide isosteres : the core unit of potent HIV-1 protease inhibitors
- Author
- GHOSH, A. K; MCKEE, S. P; THOMPSON, W. J
Merck Sharp & Dohme Research Laboratories, dep. medicinal chemistry, West Point PA 19486, United States - Source
Journal of organic chemistry. 1991, Vol 56, Num 23, pp 6500-6503 ; ref : 21 ref
- CODEN
- JOCEAH
- ISSN
- 0022-3263
- Scientific domain
- Biochemistry, molecular biology, biophysics; Organic chemistry
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Alcool secondaire Aminoalcool Composé benzénique Enantiosélectivité Hydroxyamide Mannose Stéréosélectivité Caproïque acide(2-benzyl-5-[t-butoxycarbonylamino]-4-hydroxy-6-phényl) benzylamide Furan-2-one(3-benzyl-5-[α-(t-butoxycarbonylamino) phénéthyl]-2,3,4,5-tétrahydro)
- Keyword (en)
- Secondary alcohol Aminoalcohol Benzenic compound Enantioselectivity Hydroxyamide Mannose Stereoselectivity
- Keyword (es)
- Alcohol secundario Aminoalcohol Compuesto bencénico Enantioselectividad Hidroxiamida Manosa Estereoselectividad
- Classification
- Pascal
- 001 Exact sciences and technology / 001C Chemistry / 001C03 Organic chemistry / 001C03C Preparations and properties / 001C03C03 Noncondensed benzenic compounds
- Discipline
- Organic chemistry
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 5031286
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jo00023a009 
https://dx.doi.org/10.1021/jo00023a009
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