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Potent indole- and quinoline-containing N-methyl-D-aspartate antagonists acting at the strychnine-insensitive glycine binding site

Author
BARON, B. M1 ; HARRISON, B. L; MCDONALD, I. A; MELDRUM, B. S; PALFREYMAN, M. G; SALITURO, F. G; SIEGEL, B. W; SLONE, A. L; TURNER, J. P; WHITE, H. S
[1] Marion Merrel Dow res. inst., Cincinnati OH 45215, United States
Source

The Journal of pharmacology and experimental therapeutics. 1992, Vol 262, Num 3, pp 947-956 ; ref : 1/2 p

CODEN
JPETAB
ISSN
0022-3565
Scientific domain
Pharmacology drugs
Publisher
American Society for Pharmacology and Experimental Therapeutics, Bethesda, MD
Publication country
United States
Document type
Article
Language
English
Keyword (fr)
Aminoacide excitateur Animal Antagoniste Anticonvulsivant Chimiothérapie Convulsion Encéphale Fixation biologique Glycine In vitro In vivo Mécanisme action Récepteur NMDA Récepteur glutamate Site fixation Strychnine Système nerveux central Traitement MDL 100 748 MDL 29 951 NMDA Système nerveux pathologie
Keyword (en)
Excitatory aminoacid Animal Antagonist Anticonvulsant Chemotherapy Convulsion Brain (vertebrata) Biological fixation Glycine In vitro In vivo Mechanism of action NMDA receptor Glutamate receptor Binding site Central nervous system Treatment Nervous system diseases
Keyword (es)
Aminoácido excitador Animal Antagonista Anticonvulsivante Quimioterapia Convulsión Encéfalo Fijación biológica Glicina In vitro In vivo Mecanismo acción Receptor NMDA Receptor glutámato Sitio fijación Sistema nervioso central Tratamiento Sistema nervioso patología
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02B Neuropharmacology / 002B02B06 Anticonvulsants. Antiepileptics. Antiparkinson agents

Discipline
Pharmacological treatments Psychopathology. Psychiatry. Clinical psychology
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
5604853

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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