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au.\*:("ANTHES, John C")

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Characterization of adenosine receptors in the human bladder carcinoma T24 cell lineTARA PHELPS, P; ANTHES, John C; CORRELL, Craig C et al.European journal of pharmacology. 2006, Vol 536, Num 1-2, pp 28-37, issn 0014-2999, 10 p.Article

Cloning and functional characterization of dog transient receptor potential vanilloid receptor-1 (TRPV1)PHELPS, P. Tara; ANTHES, John C; CORRELL, Craig C et al.European journal of pharmacology. 2005, Vol 513, Num 1-2, pp 57-66, issn 0014-2999, 10 p.Article

Identification of a novel 1'-[5-((3,5-dichlorobenzoyl)methylamino)-3-(3,4-dichlorophenyl)-4-(methoxyimino) pentyl]-2-oxo-(1,4'-bipiperidine) as a dual NK1/NK2 antagonistTING, Pauline C; LEE, Joe F; SHIH, Neng-Yang et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 16, pp 2125-2128, issn 0960-894XArticle

The design and synthesis of novel NK1/NK2 dual antagonistsREICHARD, Gregory A; BALL, Zachary T; ASLANIAN, Robert et al.Bioorganic & medicinal chemistry letters (Print). 2000, Vol 10, Num 20, pp 2329-2332, issn 0960-894XArticle

Reduction of CYP450 inhibition in the 4-[(1H-imidazol-4-yl)methyl]piperidine series of histamine H3 receptor antagonistsBERLIN, Michael; TING, Pauline C; DUGUMA, Luli et al.Bioorganic & medicinal chemistry letters (Print). 2006, Vol 16, Num 4, pp 989-994, issn 0960-894X, 6 p.Article

SCH 206272: a potent, orally active tachykinin NK1, NK2, and NK3 receptor antagonistANTHES, John C; CHAPMAN, Richard W; RIZZO, Charles et al.European journal of pharmacology. 2002, Vol 450, Num 2, pp 191-202, issn 0014-2999Article

Structure-activity relationships of oxime neurokinin antagonists: Oxime modificationsREICHARD, Gregory A; SPITLER, James; ASLANIAN, Robert et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 5, pp 833-836, issn 0960-894XArticle

Changes in Upper and Lower Airway Inflammation Following Administration of Mometasone Furoate in Allergen-Challenged Brown Norway RatsANTHES, John C; MCLEOD, Robbie L; KELLY, George et al.Arzneimittel-Forschung. 2009, Vol 59, Num 1, pp 13-20, issn 0004-4172, 8 p.Article

Synthesis and NK1/NK2 binding activities of a series of diacyl-substituted 2-arylpiperazinesBLYTHIN, David J; XIAO CHEN; PIWINSKI, John J et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 21, pp 3161-3165, issn 0960-894X, 5 p.Article

Tryptase-induced airway microvascular leakage in guinea pigs : involvement of tachykinins and leukotrienesGREENFEDER, Scott; SEHRING, Susan; MCHUGH, Nansie et al.European journal of pharmacology. 2001, Vol 419, Num 2-3, pp 261-267, issn 0014-2999Article

The synthesis and structure-activity relationship of 4-benzimidazolyl-piperidinylcarbonyl-piperidine analogs as histamine H3 antagonistsTING, Pauline C; LEE, Joe F; ANTHES, John C et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 17, pp 5004-5008, issn 0960-894X, 5 p.Article

Cloning and pharmacological characterization of mouse TRPV1CORRELL, Craig C; PHELPS, P. Tara; ANTHES, John C et al.Neuroscience letters. 2004, Vol 370, Num 1, pp 55-60, issn 0304-3940, 6 p.Article

Preparation of oxime dual NK1/NK2 antagonists with reduced NK3 affinityREICHARD, Gregory A; GRICE, Cheryl A; SHIH, Neng-Yang et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 17, pp 2355-2358, issn 0960-894XArticle

Synthesis and structure-activity relationships of oxime neurokinin antagonists: Discovery of potent arylamidesSHIH, Neng-Yang; ALBANESE, Margaret; WONG, Shing-Chung et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 2, pp 141-145, issn 0960-894XArticle

Novel histamine H3 receptor antagonists based on the 4-[(1H-imidazol-4-yl)methyl]piperidine scaffoldVACCARO, Wayne D; SHER, Rosy; WILLIAMS, Shirley M et al.Bioorganic & medicinal chemistry letters (Print). 2006, Vol 16, Num 2, pp 395-399, issn 0960-894X, 5 p.Article

Desloratadine inhibits constitutive and histamine-stimulated nuclear factor-κB activity consistent with inverse agonism at the histamine H1 receptorWU, Ren-Long; ANTHES, John C; KREUTNER, William et al.International archives of allergy and immunology. 2004, Vol 135, Num 4, pp 313-318, issn 1018-2438, 6 p.Article

A family of depsi-peptide fungal metabolites, as selective and competitive human tachykinin receptor (NK2) antagonists : Fermentation, isolation, physico-chemical properties, and biological activityHEGDE, Vinod R; PUAR, Mohindar S; PING DAI et al.Journal of antibiotics (Tokyo. 1968). 2001, Vol 54, Num 2, pp 125-135, issn 0021-8820Article

Spiro-piperidine azetidinones as potent TRPV1 antagonistsDONG XIAO; PALANI, Anandan; ASLANIAN, Robert et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 3, pp 783-787, issn 0960-894X, 5 p.Article

Biochemical characterization of desloratadine, a potent antagonist of the human histamine H1 receptorANTHES, John C; GILCHREST, Helen; EGAN, Robert W et al.European journal of pharmacology. 2002, Vol 449, Num 3, pp 229-237, issn 0014-2999Article

Synthesis of substituted 4(Z)-(methoxyimino)pentyl-1-piperidines as dual NK1/NK2 inhibitorsTING, Pauline C; LEE, Joe F; ANTHES, John C et al.Bioorganic & medicinal chemistry letters (Print). 2001, Vol 11, Num 4, pp 491-494, issn 0960-894XArticle

Synthesis and NK1/NK2 receptor activity of substituted-4(Z)-(methoxyimino)pentyl-1-piperazinesTING, Pauline C; LEE, Joe F; ANTHES, John C et al.Bioorganic & medicinal chemistry letters (Print). 2000, Vol 10, Num 20, pp 2333-2335, issn 0960-894XArticle

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