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Highly potent and selective chiral inhibitors of PDE5 : An illustration of Pfeiffer's ruleBUNNAGE, Mark E; MATHIAS, John P; WOOD, Anthony et al.Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 23, pp 6033-6036, issn 0960-894X, 4 p.Article

Lead diversification. Application to existing drug molecules: Mifepristone 1 and antalarmin 8ABID MASOOD, M; FARRANT, Elizabeth; MORAO, Inaki et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 1, pp 723-728, issn 0960-894X, 6 p.Article

Discovery of Potent & Selective Inhibitors of Activated Thrombin-Activatable Fibrinolysis Inhibitor for the Treatment of ThrombosisBUNNAGE, Mark E; BLAGG, Julian; EVANS, Karen et al.Journal of medicinal chemistry (Print). 2007, Vol 50, Num 24, pp 6095-6103, issn 0022-2623, 9 p.Article

Lead Diversification 2: Application to P38, gMTP and lead compoundsABID MASOOD, M; BAZIN, Marc; PEAKMAN, Torren et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 2, pp 1255-1262, issn 0960-894X, 8 p.Article

Inhalation by design: Dual pharmacology β-2 agonists/M3 antagonists for the treatment of COPDJONES, Lyn H; BALDOCK, Helen; HILTON, Laura et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 9, pp 2759-2763, issn 0960-894X, 5 p.Article

PFI-1, a Highly Selective Protein Interaction Inhibitor, Targeting BET BromodomainsPICAUD, Sarah; DA COSTA, David; BRADNER, James E et al.Cancer research (Chicago, Ill.). 2013, Vol 73, Num 11, pp 3336-3346, issn 0008-5472, 11 p.Article

Oxygenated analogues of UK-396082 as inhibitors of activated thrombin activatable fibrinolysis inhibitorOWEN, Dafydd R; BULL, David J; BUNNAGE, Mark E et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 1, pp 92-96, issn 0960-894X, 5 p.Article

The discovery of long acting β2-adrenoreceptor agonistsBROWN, Alan D; BUNNAGE, Mark E; TREVETHICK, Mike et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 14, pp 4012-4015, issn 0960-894X, 4 p.Article

Acidic triazoles as soluble guanylate cyclase stimulatorsROBERTS, Lee R; BRADLEY, Paul A; SMITH, Graham L et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 21, pp 6515-6518, issn 0960-894X, 4 p.Article

The discovery of adamantyl-derived, inhaled, long acting β2-adrenoreceptor agonistsBROWN, Alan D; BUNNAGE, Mark E; TREVETHICK, Mike et al.Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 4, pp 1280-1283, issn 0960-894X, 4 p.Article

The discovery of indole-derived long acting β2-adrenoceptor agonists for the treatment of asthma and COPDBROWN, Alan D; BUNNAGE, Mark E; WEBSTER, Rob et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 22, pp 6188-6191, issn 0960-894X, 4 p.Article

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