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au.\*:("CALVO, Margarita")

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The mechanisms of microgliosis and pain following peripheral nerve injuryCALVO, Margarita; BENNETT, David L. H.Experimental neurology (Print). 2012, Vol 234, Num 2, pp 271-282, issn 0014-4886, 12 p.Article

A clinically relevant rodent model of the HIV antiretroviral drug stavudine induced painful peripheral neuropathyWENLONG HUANG; CALVO, Margarita; KARU, Kersti et al.Pain (Amsterdam). 2013, Vol 154, Num 4, pp 560-575, issn 0304-3959, 16 p.Article

Discovery of potent, selective human granzyme B inhibitors that inhibit CTL mediated apoptosisWILLOUGHBY, Christopher A; BULL, Herbert G; GARCIA-CALVO, Margarita et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 16, pp 2197-2200, issn 0960-894XArticle

Multiple strategies for the preparation of a sulfur-35 labeled NPC1L1 radioligandSIMEONE, Joseph P; BRAUN, Matthew P; LEONE, Joseph F et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 17, pp 5033-5036, issn 0960-894X, 4 p.Article

Spiroimidazolidinone NPC1L1 inhibitors. 1: Discovery by 3D-similarity-based virtual screeningMCMASTERS, Daniel R; GARCIA-CALVO, Margarita; MAIOROV, Vladimir et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 11, pp 2965-2968, issn 0960-894X, 4 p.Article

Spiroimidazolidinone NPC1L1 inhibitors. Part 2: Structure―activity studies and in vivo efficacyHOWELL, Kobporn L; DEVITA, Robert J; GARCIA-CALVO, Margarita et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 23, pp 6929-6932, issn 0960-894X, 4 p.Article

Peptidomic profiling of human cerebrospinal fluid identifies YPRPIHPA as a novel substrate for prolylcarboxypeptidaseXUEMEI ZHAO; SOUTHWICK, Katie; GARCIA-CALVO, Margarita et al.Proteomics (Weinheim. Print). 2010, Vol 10, Num 15, pp 2882-2886, issn 1615-9853, 5 p.Article

A new class of prolylcarboxypeptidase inhibitors, Part 2: The aminocyclopentanesGRAHAM, Thomas H; WENSHENGLIU; HUAIBING HE et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 8, pp 2818-2822, issn 0960-894X, 5 p.Article

Discovery of benzimidazole pyrrolidinyl amides as prolylcarboxypeptidase inhibitorsSHEN, Hong C; DING, Fa-Xiang; BHATT, Urmi R et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 5, pp 1299-1305, issn 0960-894X, 7 p.Article

Discovery of a new class of potent prolylcarboxypeptidase inhibitors derived from alanineZHICAI WU; CANGMING YANG; LASSMAN, Mike E et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 4, pp 1774-1778, issn 0960-894X, 5 p.Article

Discovery of novel aspartyl ketone dipeptides as potent and selective caspase-3 inhibitorsYONGXIN HAN; GIROUX, André; RASPER, Dita M et al.Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 3, pp 805-808, issn 0960-894X, 4 p.Article

Discovery of benzodihydroisofurans as novel, potent, bioavailable and brain-penetrant prolylcarboxypeptidase inhibitorsSHEN, Hong C; DING, Fa-Xiang; BHATT, Urmi R et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 4, pp 1550-1556, issn 0960-894X, 7 p.Article

Discovery of aminoheterocycles as potent and brain penetrant prolylcarboxypeptidase inhibitorsZHICAI WU; CANGMING YANG; GARCIA-CALVO, Margarita M et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 4, pp 1727-1730, issn 0960-894X, 4 p.Article

The discovery of non-benzimidazole and brain-penetrant prolylcarboxypeptidase inhibitorsGRAHAM, Thomas H; SHEN, HongC; GARCIA-CALVO, Margarita et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 1, pp 658-665, issn 0960-894X, 8 p.Article

A new class of prolylcarboxypeptidase inhibitors, Part 1: Discovery and evaluationGRAHAM, Thomas H; WENSHENG LIU; GORSKI, Judith N et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 8, pp 2811-2817, issn 0960-894X, 7 p.Article

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