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au.\*:("FERANDIN, Yoan")

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An integrated computational approach to the phenomenon of potent and selective inhibition of aurora kinases B and C by a series of 7-substituted indirubinsMYRIANTHOPOULOS, Vassilios; MAGIATIS, Prokopios; FERANDIN, Yoan et al.Journal of medicinal chemistry (Print). 2007, Vol 50, Num 17, pp 4027-4037, issn 0022-2623, 11 p.Article

Synthesis and biological activities of aminopyrimidyl-indoles structurally related to meridianinsAKUE-GEDU, Rufine; DEBITON, Eric; FERANDIN, Yoan et al.Bioorganic & medicinal chemistry. 2009, Vol 17, Num 13, pp 4420-4424, issn 0968-0896, 5 p.Article

3'-substituted 7-halogenoindirubins, a new class of cell death inducing agentsFERANDIN, Yoan; BETTAYEB, Karima; KRITSANIDA, Marina et al.Journal of medicinal chemistry (Print). 2006, Vol 49, Num 15, pp 4638-4649, issn 0022-2623, 12 p.Article

Design, synthesis, and testing of an 6-0-linked series of benzimidazole based inhibitors of CDK5/p25JAIN, Prashi; FLAHERTY, Patrick T; SHUYAN YI et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 1, pp 359-373, issn 0968-0896, 15 p.Article

Development of 5-benzylpaullones and paullone-9-carboxylic acid alkyl esters as selective inhibitors of mitochondrial malate dehydrogenase (mMDH)BECKER, Anja; KOHFELD, Simone; LADER, Annette et al.European journal of medicinal chemistry. 2010, Vol 45, Num 1, pp 335-342, issn 0223-5234, 8 p.Article

Synthesis of novel 5-substituted indirubins as protein kinases inhibitorsBEAUCHARD, Anne; FERANDIN, Yoan; FRERE, Stéphane et al.Bioorganic & medicinal chemistry. 2006, Vol 14, Num 18, pp 6434-6443, issn 0968-0896, 10 p.Article

Meriolins (3-(Pyrimidin-4-yl)-7-azaindoles) : Synthesis, Kinase Inhibitory Activity, Cellular Effects, and Structure of a CDK2/Cyclin A/Meriolin ComplexECHALIER, Aude; BETTAYEB, Karima; JOSEPH, Benoit et al.Journal of medicinal chemistry (Print). 2008, Vol 51, Num 4, pp 737-751, issn 0022-2623, 15 p.Article

Pyrazolo[1,5-a]-1,3,5-triazine as a Purine Bioisostere : Access to Potent Cyclin-Dependent Kinase Inhibitor (R)-Roscovitine AnaloguePOPOWYCZ, Florence; FOUMET, Guy; BERNARD, Philippe et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 3, pp 655-663, issn 0022-2623, 9 p.Article

9-Cyano-1-azapaullone (Cazpaullone), a Glycogen Synthase Kinase-3 (GSK-3) Inhibitor Activating Pancreatic β Cell Protection and ReplicationSTUKENBROCK, Hendrik; MUSSMANN, Rainer; MEIJER, Laurent et al.Journal of medicinal chemistry (Print). 2008, Vol 51, Num 7, pp 2196-2207, issn 0022-2623, 12 p.Article

Synthesis and kinase inhibitory activity of novel substituted indigoidsBEAUCHARD, Anne; LABORIE, Hélène; ROUILLARD, Hervé et al.Bioorganic & medicinal chemistry. 2009, Vol 17, Num 17, pp 6257-6263, issn 0968-0896, 7 p.Article

Soluble 3',6-Substituted Indirubins with Enhanced Selectivity toward Glycogen Synthase Kinase -3 Alter Circadian PeriodVOUGOGIANNOPOULOU, Konstantina; FERANDIN, Yoan; MEIJER, Laurent et al.Journal of medicinal chemistry (Print). 2008, Vol 51, Num 20, pp 6421-6431, issn 0022-2623, 11 p.Article

Roscovitine-Derived, Dual-Specificity Inhibitors of Cyclin-Dependent Kinases and Casein Kinases 1OUMATA, Nassima; BETTAYEB, Karima; MEIJER, Laurent et al.Journal of medicinal chemistry (Print). 2008, Vol 51, Num 17, pp 5229-5242, issn 0022-2623, 14 p.Article

Meriolins, a new class of cell death -Inducing kinase inhibitors with enhanced selectivity for cyclin-dependent kinasesBETTAYEB, Karima; TIRADE, Oscar M; LIGER, Francois et al.Cancer research (Baltimore). 2007, Vol 67, Num 17, pp 8325-8334, issn 0008-5472, 10 p.Article

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