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Overcoming Persistent Dependency on Androgen Signaling after Progression to Castration-Resistant Prostate CancerYAMAOKA, Masuo; HARA, Takahito; KUSAKA, Masami et al.Clinical cancer research (Print). 2010, Vol 16, Num 17, pp 4319-4324, issn 1078-0432, 6 p.Article

Novel benzimidazole derivatives selectively inhibit endothelial cell growth and suppress angiogenesis in vitro and in vivoHORI, Akira; IMAEDA, Yasuhiro; KUBO, Keiji et al.Cancer letters. 2002, Vol 183, Num 1, pp 53-60, issn 0304-3835Article

Possible role of adaptive mutation in resistance to antiandrogen in prostate cancer cellsHARA, Takahito; KOUNO, Jin; NAKAMURA, Kazuyo et al.The Prostate. 2005, Vol 65, Num 3, pp 268-275, issn 0270-4137, 8 p.Article

Enhanced androgen receptor signaling correlates with the androgen-refractory growth in a newly established MDA PCa 2b-hr human prostate cancer cell sublineHARA, Takahito; NAKAMURA, Kazuyo; ARAKI, Hideo et al.Cancer research (Baltimore). 2003, Vol 63, Num 17, pp 5622-5628, issn 0008-5472, 7 p.Article

A Novel Androgen-Dependent Prostate Cancer Xenograft Model Derived From Skin Metastasis of a Japanese PatientKIMURA, Takahiro; KIYOTA, Hiroshi; NAKATA, Daisuke et al.The Prostate. 2009, Vol 69, Num 15, pp 1660-1667, issn 0270-4137, 8 p.Article

Design, synthesis, and biological evaluation of 4-phenylpyrrole derivatives as novel androgen receptor antagonistsYAMAMOTO, Satoshi; MATSUNAGA, Nobuyuki; FURUYA, Shuichi et al.Bioorganic & medicinal chemistry. 2012, Vol 20, Num 1, pp 422-434, issn 0968-0896, 13 p.Article

Novel mutations of androgen receptor: A possible mechanism of bicalutamide withdrawal syndromeHARA, Takahito; MIYAZAKI, Jun-Ichi; ARAKI, Hideo et al.Cancer research (Baltimore). 2003, Vol 63, Num 1, pp 149-153, issn 0008-5472, 5 p.Article

Suppression of a pituitary-ovarian axis by chronic oral administration of a novel nonpeptide gonadotropin-releasing hormone antagonist, TAK-013, in cynomolgus monkeysHARA, Takahito; ARAKI, Hideo; KUSAKA, Masami et al.The Journal of clinical endocrinology and metabolism. 2003, Vol 88, Num 4, pp 1697-1704, issn 0021-972X, 8 p.Article

2-Acylamino-4,6-diphenylpyridine derivatives as novel GPR54 antagonists with good brain exposure and in vivo efficacy for plasma LH level in male ratsKOBAYASHI, Toshitake; SASAKI, Satoshi; BABA, Atsuo et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 14, pp 5157-5171, issn 0968-0896, 15 p.Article

Chronic Administration of the Metastin/Kisspeptin Analog KISS1-305 or the Investigational Agent TAK-448 Suppresses Hypothalamic Pituitary Gonadal Function and Depletes Plasma Testosterone in Adult Male RatsMATSUI, Hisanori; TANAKA, Akira; KUSAKA, Masami et al.Endocrinology (Philadelphia). 2012, Vol 153, Num 11, pp 5297-5308, issn 0013-7227, 12 p.Article

Discovery of orteronel (TAK-700), a naphthylmethylimidazole derivative, as a highly selective 17,20-lyase inhibitor with potential utility in the treatment of prostate cancerKAKU, Tomohiro; HITAKA, Takenori; ASAHI, Satoru et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 21, pp 6383-6399, issn 0968-0896, 17 p.Article

C17,20-lyase inhibitors. Part 2: Design, synthesis and structure-activity relationships of (2-naphthylmethyl)-1H-imidazoles as novel C17,20-lyase inhibitorsMATSUNAGA, Nobuyuki; KAKU, Tomohiro; OJIDA, Akio et al.Bioorganic & medicinal chemistry. 2004, Vol 12, Num 16, pp 4313-4336, issn 0968-0896, 24 p.Article

17,20-Lyase inhibitors. Part 3: Design, synthesis, and structure-activity relationships of biphenylylmethylimidazole derivatives as novel 17,20-lyase inhibitorsKAKU, Tomohiro; TSUJIMOTO, Saori; MATSUNAGA, Nobuyuki et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 7, pp 2428-2442, issn 0968-0896, 15 p.Article

17,20-Lyase inhibitors. Part 4: Design, synthesis and structure―activity relationships of naphthylmethylimidazole derivatives as novel 17,20-lyase inhibitorsKAKU, Tomohiro; MATSUNAGA, Nobuyuki; OJIDA, Akio et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 5, pp 1751-1770, issn 0968-0896, 20 p.Article

C17,20-Lyase inhibitors I. Structure-based de novo design and SAR study of C17,20-lyase inhibitorsMATSUNAGA, Nobuyuki; KAKU, Tomohiro; TASAKA, Akihiro et al.Bioorganic & medicinal chemistry. 2004, Vol 12, Num 9, pp 2251-2273, issn 0968-0896, 23 p.Article

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