The cultural sublime and the temporal dimension of media: The case of child murderer Marc DutrouxLEURS, Rob.International journal of cultural studies (Print). 2009, Vol 12, Num 4, pp 395-414, issn 1367-8779, 20 p.Article

Delineation of receptor-ligand interactions at the human histamine H₁ receptor by a combined approach of site-directed mutagenesis and computational techniques - or - how to bind the H₁ receptorJONGEJAN, Aldo; LEURS, Rob.Archiv der Pharmazie (Weinheim). 2005, Vol 338, Num 5-6, pp 248-259, issn 0365-6233, 12 p.Article

The histamine H₃ receptor (a target for new drugs)Leurs, Rob; Timmerman, Henk.Pharmacochemistry library. 1998, issn 0165-7208, isbn 0-444-82936-9, XI, 291 p, isbn 0-444-82936-9Book

Activation of peripheral and spinal histamine H₃ receptors inhibits formalin-induced inflammation and nociception, respectivelyCANNON, Keri E; LEURS, Rob; HOUGH, Lindsay B et al.Pharmacology, biochemistry and behavior. 2007, Vol 88, Num 1, pp 122-129, issn 0091-3057, 8 p.Article

Role of H₃-receptor-mediated signaling in anxiety and cognition in wild-type and Apoe^-/- miceBONGERS, Gerald; LEURS, Rob; ROBERTSON, Jennifer et al.Neuropsychopharmacology (New York, NY). 2004, Vol 29, Num 3, pp 441-449, issn 0893-133X, 9 p.Article

Modulation of histamine H₂ receptor signalling by G-protein-coupled receptor kinase 2 and 3RODRIGUEZ-PENA, Maria Sol; TIMMERMAN, Henk; LEURS, Rob et al.British journal of pharmacology. 2000, Vol 131, Num 8, pp 1707-1715, issn 0007-1188Article

Major advances in the development of histamine H₄ receptor ligandsSMITS, Rogier A; LEURS, Rob; DE ESCH, Iwan J. P et al.Drug discovery today. 2009, Vol 14, Num 15-16, pp 745-753, issn 1359-6446, 9 p.Article

G protein-coupled receptors: walking hand-in-hand, talking hand-in-hand?VISCHER, Henry F; WATTS, Anne O; NIJMEIJER, Saskia et al.British journal of pharmacology. 2011, Vol 163, Num 2, pp 246-260, issn 0007-1188, 15 p.Article

The role of cytomegalovirus-encoded homologs of G protein-coupled receptors and chemokines in manipulation of and evasion from the immune systemVINK, Cornelis; SMIT, Martine J; LEURS, Rob et al.Journal of clinical virology. 2001, Vol 23, Num 1-2, pp 43-55, issn 1386-6532Article

Antiinflammatory and antinociceptive effects of the selective histamine H₄-receptor antagonists JNJ7777120 and VUF6002 in a rat model of carrageenan-induced acute inflammationCORUZZI, Gabriella; ADAMI, Maristella; GUAITA, Elena et al.European journal of pharmacology. 2007, Vol 563, Num 1-3, pp 240-244, issn 0014-2999, 5 p.Article

Molecular aspects of the histamine H₃ receptorBONGERS, Gerold; BAKKER, Remko A; LEURS, Rob et al.Biochemical pharmacology. 2007, Vol 73, Num 8, pp 1195-1204, issn 0006-2952, 10 p.Article

Histamine H₃ receptor antagonists reach out for the clinicCELANIRE, Sylvain; WIJTMANS, Maikel; TALAGA, Patrice et al.Drug discovery today. 2005, Vol 10, Num 23-24, pp 1613-1627, issn 1359-6446, 15 p.Article

Transforming fragments into candidates: small becomes big in medicinal chemistryDE KLOE, Gerdien E; BAILEY, David; LEURS, Rob et al.Drug discovery today. 2009, Vol 14, Num 13-14, pp 630-646, issn 1359-6446, 17 p.Article

A locked-on, constitutively active mutant of the adenosine A₁ receptorDE LIGT, Rianne A. F; RIVKEES, Scott A; LORENZEN, Anna et al.European journal of pharmacology. 2005, Vol 510, Num 1-2, pp 1-8, issn 0014-2999, 8 p.Article

Selective histamine H₃ and H₄ receptor agonists exert opposite effects against the gastric lesions induced by HCl in the rat stomachCORUZZI, Gabriella; ADAMI, Maristella; POZZOLI, Cristina et al.European journal of pharmacology. 2011, Vol 669, Num 1-3, pp 121-127, issn 0014-2999, 7 p.Article

Fragment based lead discovery of small molecule inhibitors for the EPHA4 receptor tyrosine kinaseVAN LINDEN, Oscar P. J; FARENC, Carine; ZOUTMAN, Willem H et al.European journal of medicinal chemistry. 2012, Vol 47, pp 493-500, issn 0223-5234, 8 p.Article

CXCR3 antagonists: Quaternary ammonium salts equipped with biphenyl-and polycycloaliphatic-anchorsWIJTMANS, Maikel; VERZIJL, Dennis; BERGMANS, Serge et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 11, pp 3384-3393, issn 0968-0896, 10 p.Article

Identification of novel allosteric nonpeptidergic inhibitors of the human cytomegalovirus-encoded chemokine receptor US28VISCHER, Henry F; HULSHOF, Janneke W; HULSCHER, Saskia et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 2, pp 675-688, issn 0968-0896, 14 p.Article

4-Benzyl-lH-imidazoles with Oxazoline Termini as Histamine H₃ Receptor AgonistsWIJTMANS, Maikel; CELANIRE, Sylvain; LEBON, Florence et al.Journal of medicinal chemistry (Print). 2008, Vol 51, Num 10, pp 2944-2953, issn 0022-2623, 10 p.Article

Characterization of the histamine H₄ receptor binding site. Part 1. Synthesis and pharmacological evaluation of dibenzodiazepine derivativesSMITS, Rogier A; LIM, Herman D; STEGINK, Bart et al.Journal of medicinal chemistry (Print). 2006, Vol 49, Num 15, pp 4512-4516, issn 0022-2623, 5 p.Article

Mutational analysis of the histamine H₁-receptor binding pocket of histaprodifensBRUYSTERS, Martijn; PERTZ, Heinz H; TEUNISSEN, Aloys et al.European journal of pharmacology. 2004, Vol 487, Num 1-3, pp 55-63, issn 0014-2999, 9 p.Article

Synthesis and structure-activity relationships of indole and benzimidazole piperazines as histamine H₄ receptor antagonistsTERZIOGLU, Nalan; VAN RIJN, Richard M; BAKKER, Remko A et al.Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 21, pp 5251-5256, issn 0960-894X, 6 p.Article

Development of a pharmacophore model for histamine H₃ receptor antagonists, using the newly developed molecular modeling program SLATEDE ESCH, Iwan J. P; MILLS, James E. J; TIMMERMAN, Henk et al.Journal of medicinal chemistry (Print). 2001, Vol 44, Num 11, pp 1666-1674, issn 0022-2623Article

Strain-dependent effects of the histamine H₄ receptor antagonist JNJ7777120 in a murine model of acute skin inflammationCORUZZI, Gabriella; POZZOLI, Cristina; ADAMI, Maristella et al.Experimental dermatology. 2012, Vol 21, Num 1, pp 32-37, issn 0906-6705, 6 p.Article

Structure-based design, synthesis and structure―activity relationships of dibenzosuberyl- and benzoate-substituted tropines as ligands for acetylcholine-binding proteinEDINK, Ewald; AKDEMIR, Atilla; JANSEN, Chimed et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 3, pp 1448-1454, issn 0960-894X, 7 p.Article