The growing impact of click chemistry on drug discovery = L'impact de la chimie sur la découverte de médicamentsKOLB, Hartmuth C; SHARPLESS, K. Barry.Drug discovery today. 2003, Vol 8, Num 24, pp 1128-1137, issn 1359-6446, 10 p.Article

Why is tetrazole formation by addition of azide to organic nitriles catalyzed by zinc(II) salts?HIMO, Fahmi; DEMKO, Zachary P; NOODLEMAN, Louis et al.Journal of the American Chemical Society. 2003, Vol 125, Num 33, pp 9983-9987, issn 0002-7863, 5 p.Article

Mechanisms of tetrazole formation by addition of azide to nitrilesHIMO, Fahmi; DEMKO, Zachary P; NOODLEMAN, Louis et al.Journal of the American Chemical Society. 2002, Vol 124, Num 41, pp 12210-12216, issn 0002-7863, 7 p.Article

Nucleophilic substitution by Grignard reagents on sulfur mustardsCONVERSO, Antonella; SAAIDI, Pierre-Loïc; SHARPLESS, K. Barry et al.Journal of organic chemistry. 2004, Vol 69, Num 21, pp 7336-7339, issn 0022-3263, 4 p.Article

The allylic azide rearrangement : Achieving selectivityFELDMAN, Alina K; COLASSON, Benott; SHARPLESS, K. Barry et al.Journal of the American Chemical Society. 2005, Vol 127, Num 39, pp 13444-13445, issn 0002-7863, 2 p.Article

Ruthenium-catalyzed cycloaddition of alkynes and organic azidesLI ZHANG; XINGUO CHEN; PENG XUE et al.Journal of the American Chemical Society. 2005, Vol 127, Num 46, pp 15998-15999, issn 0002-7863, 2 p.Article

In situ click chemistry: Enzyme inhibitors made to their own specificationsMANETSCH, Roman; KRASINSKI, Antoni; RADIC, Zoran et al.Journal of the American Chemical Society. 2004, Vol 126, Num 40, pp 12809-12818, issn 0002-7863, 10 p.Article

Design and synthesis via click chemistry of 8,9-anhydroerythromycin a 6,9-hemiketal analogues with anti-MRSA and -VRE activitySUGAWARA, Akihiro; SUNAZUKA, Toshiaki; HIROSE, Tomoyasu et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 22, pp 6340-6344, issn 0960-894X, 5 p.Article

Rapid discovery and structure-activity profiling of novel inhibitors of human immunodeficiency virus type 1 protease enabled by the copper(I)-catalyzed synthesis of 1,2,3-triazoles and their further functionalizationWHITING, Matthew; TRIPP, Jonathan C; LIN, Ying-Chuan et al.Journal of medicinal chemistry (Print). 2006, Vol 49, Num 26, pp 7697-7710, issn 0022-2623, 14 p.Article

Bisaryloxime ethers as potent inhibitors of transthyretin amyloid fibril formationJOHNSON, Steven M; PETRASSI, H. Michael; KELLY, Jeffery W et al.Journal of medicinal chemistry (Print). 2005, Vol 48, Num 5, pp 1576-1587, issn 0022-2623, 12 p.Article

Role of architecture and molecular weight in the formation of tailor-made ultrathin multilayers using dendritic macromolecules and click chemistryVESTBERG, Robert; MALKOCH, Michael; KADE, Matthew et al.Journal of polymer science. Part A. Polymer chemistry. 2007, Vol 45, Num 14, pp 2835-2846, issn 0887-624X, 12 p.Article

Bioconjugation by copper(I)-catalyzed azide-alkyne [3 + 2] cycloadditionQIAN WANG; CHAN, Timothy R; HILGRAF, Robert et al.Journal of the American Chemical Society. 2003, Vol 125, Num 11, pp 3192-3193, issn 0002-7863, 2 p.Article

A potent and highly selective inhibitor of human α-1,3-fucosyltransferase via click chemistryLEE, Lac V; MITCHELL, Michael L; HUANG, Shih-Jung et al.Journal of the American Chemical Society. 2003, Vol 125, Num 32, pp 9588-9589, issn 0002-7863, 2 p.Article

Automated Docking with Protein Flexibility in the Design of Femtomolar Click Chemistry Inhibitors of AcetylcholinesteraseMORRIS, Garrett M; GREEN, Luke G; RADIC, Zoran et al.Journal of chemical information and modeling. 2013, Vol 53, Num 4, pp 898-906, issn 1549-9596, 9 p.Article

A Sulfilimine Bond Identified in Collagen IVVANACORE, Roberto; HAM, Amy-Joan L; VOEHLER, Markus et al.Science (Washington, D.C.). 2009, Vol 325, Num 5945, pp 1230-1234, issn 0036-8075, 5 p.Article

Synthesis and Electrochemistry of 2-Ethenyl and 2-Ethanyl Derivatives of 5-Nitroimidazole and Antimicrobial Activity against Giardia lambliaVALDEZ, Carlos A; TRIPP, Jonathan C; GILLIN, Frances D et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 13, pp 4038-4053, issn 0022-2623, 16 p.Article

Mechanistic Studies on the Cu-Catalyzed Three-Component Reactions of Sulfonyl Azides, 1-Alkynes and Amines, Alcohols, or Water : Dichotomy via a Common PathwayEUN JEONG YOO; AHLQUIST, Marten; BAE, Imhyuck et al.Journal of organic chemistry. 2008, Vol 73, Num 14, pp 5520-5528, issn 0022-3263, 9 p.Article

Click chemistry in materials synthesis. III. Metal-adhesive polymers from Cu(I)-catalyzed azide-alkyne cycloadditionYI LIU; DIAZ, David D; ACCURSO, Adrian A et al.Journal of polymer science. Part A. Polymer chemistry. 2007, Vol 45, Num 22, pp 5182-5189, issn 0887-624X, 8 p.Article

Copper(I)-catalyzed synthesis of azoles. DFT study predicts unprecedented reactivity and intermediatesHIMO, Fahmi; LOVELL, Timothy; HILGRAF, Robert et al.Journal of the American Chemical Society. 2005, Vol 127, Num 1, pp 210-216, issn 0002-7863, 7 p.Article

In situ selection of lead compounds by click chemistry : Target-guided optimization of acetylcholinesterase inhibitorsKRASINSKI, Antoni; RADIC, Zoran; MANETSCH, Roman et al.Journal of the American Chemical Society. 2005, Vol 127, Num 18, pp 6686-6692, issn 0002-7863, 7 p.Article

Click chemistry in materials synthesis. 1. Adhesive polymers from copper-catalyzed azide-alkyne cycloadditionDIAZ, David D; PUNNA, Sreenivas; HOLZER, Philipp et al.Journal of polymer science. Part A. Polymer chemistry. 2004, Vol 42, Num 17, pp 4392-4403, issn 0887-624X, 12 p.Article