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au.\*:("SHIH, Neng-Yang")

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Results 1 to 25 of 47

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Potent aza-peptide derived inhibitors of HCV NS3 proteaseVENKATRAMAN, Srikanth; WANLI WU; SHIH, Neng-Yang et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 16, pp 4760-4763, issn 0960-894X, 4 p.Article

Benzimidazole-substituted (3-phenoxypropyl)amines as histamine H3 receptor ligandsASLANIAN, Robert; XIAOHONG ZHU; VACCARO, Henry A et al.Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 18, pp 5032-5036, issn 0960-894X, 5 p.Article

The design and synthesis of novel NK1/NK2 dual antagonistsREICHARD, Gregory A; BALL, Zachary T; ASLANIAN, Robert et al.Bioorganic & medicinal chemistry letters (Print). 2000, Vol 10, Num 20, pp 2329-2332, issn 0960-894XArticle

Synthesis and NK1/NK2 binding activities of a series of diacyl-substituted 2-arylpiperazinesBLYTHIN, David J; XIAO CHEN; PIWINSKI, John J et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 21, pp 3161-3165, issn 0960-894X, 5 p.Article

Synthesis of substituted 4(Z)-(methoxyimino)pentyl-1-piperidines as dual NK1/NK2 inhibitorsTING, Pauline C; LEE, Joe F; ANTHES, John C et al.Bioorganic & medicinal chemistry letters (Print). 2001, Vol 11, Num 4, pp 491-494, issn 0960-894XArticle

Synthesis and NK1/NK2 receptor activity of substituted-4(Z)-(methoxyimino)pentyl-1-piperazinesTING, Pauline C; LEE, Joe F; ANTHES, John C et al.Bioorganic & medicinal chemistry letters (Print). 2000, Vol 10, Num 20, pp 2333-2335, issn 0960-894XArticle

Biaryl substituted hydantoin compounds as TACE inhibitorsWENSHENG YU; LING TONG; RIZVI, Razia et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 17, pp 5286-5289, issn 0960-894X, 4 p.Article

Novel TNF-α converting enzyme (TACE) inhibitors as potential treatment for inflammatory diseasesGIRIJAVALLABHAN, Vinay M; LEI CHEN; PIWINSKI, John J et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 24, pp 7283-7287, issn 0960-894X, 5 p.Article

Preparation of oxime dual NK1/NK2 antagonists with reduced NK3 affinityREICHARD, Gregory A; GRICE, Cheryl A; SHIH, Neng-Yang et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 17, pp 2355-2358, issn 0960-894XArticle

Synthesis and structure-activity relationships of oxime neurokinin antagonists: Discovery of potent arylamidesSHIH, Neng-Yang; ALBANESE, Margaret; WONG, Shing-Chung et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 2, pp 141-145, issn 0960-894XArticle

5-Benzothiazole substituted pyrimidine derivatives as HCV replication (replicase) inhibitorsARASAPPAN, Ashok; BENNETT, Frank; PINTO, Patrick et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 9, pp 3229-3234, issn 0960-894X, 6 p.Article

Discovery and SAR of hydantoin TACE inhibitorsWENSHENG YU; ZHUYAN GUO; LAVEY, Brian J et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 6, pp 1877-1880, issn 0960-894X, 4 p.Article

Optimization of triaryl bis-sulfones as cannabinoid-2 receptor ligandsLAVEY, Brian J; KOZLOWSKI, Joseph A; JIE WU et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 13, pp 3760-3764, issn 0960-894X, 5 p.Article

Discovery of a highly potent series of oxazole-based phosphodiesterase 4 inhibitorsKUANG, Rongze; SHUE, Ho-Jane; ASLANIAN, Robert et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 18, pp 5150-5154, issn 0960-894X, 5 p.Article

Cyclic urea derivatives as potent NK1 selective antagonistsSHUE, Ho-Jane; XIAO CHEN; PIWINSKI, John J et al.Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 17, pp 3896-3899, issn 0960-894X, 4 p.Article

Reduction of CYP450 inhibition in the 4-[(1H-imidazol-4-yl)methyl]piperidine series of histamine H3 receptor antagonistsBERLIN, Michael; TING, Pauline C; DUGUMA, Luli et al.Bioorganic & medicinal chemistry letters (Print). 2006, Vol 16, Num 4, pp 989-994, issn 0960-894X, 6 p.Article

The synthesis of substituted bipiperidine amide compounds as CCR3 ligands : Antagonists versus agonistsTING, Pauline C; UMLAND, Shelby P; YUNTAO WAN et al.Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 12, pp 3020-3023, issn 0960-894X, 4 p.Article

8-Methoxyquinolines as PDE4 inhibitorsBILLAH, Motasim; BUCKLEY, George M; MINNICOZZI, Michael et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 12, pp 1617-1619, issn 0960-894XArticle

SCH 206272: a potent, orally active tachykinin NK1, NK2, and NK3 receptor antagonistANTHES, John C; CHAPMAN, Richard W; RIZZO, Charles et al.European journal of pharmacology. 2002, Vol 450, Num 2, pp 191-202, issn 0014-2999Article

Structure-activity relationships of oxime neurokinin antagonists: Oxime modificationsREICHARD, Gregory A; SPITLER, James; ASLANIAN, Robert et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 5, pp 833-836, issn 0960-894XArticle

Synthesis and profile of SCH351591, a novel PDE4 inhibitorBILLAH, Motasim; COOPER, Nicola; KENDALL, Hannah J et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 12, pp 1621-1623, issn 0960-894XArticle

The synthesis of substituted fluorenes as novel non-imidazole histamine H3 inhibitorsTING, Pauline C; LEE, Joe F; ALBANESE, Margaret M et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 18, pp 2643-2646, issn 0960-894XArticle

II. Novel HCV NS5B polymerase inhibitors: Discovery of indole C2 acyl sulfonamidesANILKUMAR, Gopinadhan N; SELYUTIN, Oleg; LESBURG, Charles A et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 1, pp 713-717, issn 0960-894X, 5 p.Article

Novel substituted pyrimidines as HCV replication (replicase) inhibitorsKWONG, Cecil D; CLARK, Jeremy L; SHIH, Neng-Yang et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 2, pp 1160-1164, issn 0960-894X, 5 p.Article

2-(2-Aminothiazol-4-yl)pyrrolidine-based tartrate diamides as potent, selective and orally bioavailable TACE inhibitorsCHAOYANG DAI; DANSU LI; ZHUYAN GUO et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 10, pp 3172-3176, issn 0960-894X, 5 p.Article

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