Tetrahydroindolizinone NK₁ antagonistsJIANMING BAO; HUAGANG LU; MILLS, Sander G et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 7, pp 2354-2358, issn 0960-894X, 5 p.Article

Behavioral and Neurochemical Alterations in Mice Deficient in Anaplastic Lymphoma Kinase Suggest Therapeutic Potential for Psychiatric IndicationsBILSLAND, James G; WHEELDON, Alan; WHITING, Paul et al.Neuropsychopharmacology (New York, NY). 2008, Vol 33, Num 3, pp 685-700, issn 0893-133X, 16 p.Article

The discovery of potent, selective, and orally bioavailable hNK₁ antagonists derived from pyrrolidineLIN, Peter; LEHUA CHANG; KURTZ, Marc M et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 18, pp 5191-5198, issn 0960-894X, 8 p.Article

Pyrrolidine-carboxamides and oxadiazoles as potent hNK₁ antagonistsYOUNG, Jonathan R; EID, Ronsar; TURNER, Cherilyn et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 19, pp 5310-5315, issn 0960-894X, 6 p.Article

NK₁ antagonists based on seven membered lactam scaffoldsELLIOTT, Jason M; CARLSON, Emma J; WHEELDON, Alan et al.Bioorganic & medicinal chemistry letters (Print). 2006, Vol 16, Num 11, pp 2929-2932, issn 0960-894X, 4 p.Article

Synthesis and structure-activity relationships of 8-azabicyclo[3.2.1]octane benzylamine NK₁ antagonistsTHOMSON, Christopher G; CARLSON, Emma; CHICCHI, Gary G et al.Bioorganic & medicinal chemistry letters (Print). 2006, Vol 16, Num 4, pp 811-814, issn 0960-894X, 4 p.Article

UDP-glucose modulates gastric function through P2Y₁₄ receptor-dependent and -independent mechanismsBASSIL, Anna K; BOURDU, Sophie; LATCHAM, Judith et al.American journal of physiology. Gastrointestinal and liver physiology. 2009, Vol 59, Num 4, issn 0193-1857, G923-G930Article

1-Phenyl-8-azabicyclo[3.2.1]octane ethers : A novel series of neurokinin (NK₁) antagonistsHUSCROFT, Ian T; CARLSON, Emma J; CHICCHI, Gary G et al.Bioorganic & medicinal chemistry letters (Print). 2006, Vol 16, Num 7, pp 2008-2012, issn 0960-894X, 5 p.Article

Inhibition of acute nociceptive responses in rat spinal cord by a bradykinin B₁ receptor antagonistCONLEY, Rachel K; WHEELDON, Alan; WEBB, Janine K et al.European journal of pharmacology. 2005, Vol 527, Num 1-3, pp 44-51, issn 0014-2999, 8 p.Article

Substituted fused bicyclic pyrrolizinones as potent, orally bioavailable hNK₁ antagonistsMORRIELLO, Gregori J; MILLS, Sander G; XINCHUN TONG et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 6, pp 2007-2012, issn 0960-894X, 6 p.Article

Fused tricyclic pyrrolizinones that exhibit pseudo-irreversible blockade of the NK₁ receptorMORRIELLO, Gregori J; CHICCHI, Gary; TOWNSON, Karen et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 19, pp 5925-5932, issn 0960-894X, 8 p.Article

Potent, Brain-Penetrant, Hydroisoindoline-Based Human Neurokinin-1 Receptor AntagonistsJINLONG JIANG; BUNDA, Jaime L; TSCHIRRET-GUTH, Richard et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 9, pp 3039-3046, issn 0022-2623, 8 p.Article

Fused bicyclic pyrrolizinones as new scaffolds for human NK₁antagonistsMORRIELLO, Gregori J; DEVITA, Robert J; CARLSON, Emma et al.Bioorganic & medicinal chemistry. 2008, Vol 16, Num 5, pp 2156-2170, issn 0968-0896, 15 p.Article