CANNABINOID RECEPTOR CB1 ANTAGONISTS: STATE OF THE ART AND CHALLENGESBIFULCO, Maurizio; SANTORO, Antonietta; LAEZZA, Chiara et al.Vitamins and hormones. 2009, Vol 81, pp 159-189, issn 0083-6729, 31 p.Article

Peripheral cannabinoid CB₁ receptors inhibit evoked responses of nociceptive neurones in vivoKELLY, Sara; DONALDSON, Lucy F.European journal of pharmacology. 2008, Vol 586, Num 1-3, pp 160-163, issn 0014-2999, 4 p.Article

The analgesic activity of paracetamol is prevented by the blockade of cannabinoid CB₁ receptorsOTTANI, Alessandra; LEONE, Sheila; SANDRINI, Maurizio et al.European journal of pharmacology. 2006, Vol 531, Num 1-3, pp 280-281, issn 0014-2999, 2 p.Article

Pharmacological characterization of the cannabinoid CB₁ receptor PET ligand ortholog, [³H]MePPEPSUTER, Todd M; CHESTERFIELD, Amy K; CHUN BAO et al.European journal of pharmacology. 2010, Vol 649, Num 1-3, pp 44-50, issn 0014-2999, 7 p.Article

OPPOSITE ACTION OF HIPPOCAMPAL CB1 RECEPTORS IN MEMORY RECONSOLIDATION AND EXTINCTIONDE OLIVEIRA ALVARES, L; PASQUALINI GENRO, B; DIEHL, F et al.Neuroscience. 2008, Vol 154, Num 4, pp 1648-1655, issn 0306-4522, 8 p.Article

F200A substitution in the third transmembrane helix of human cannabinoid CB₁ receptor converts AM2233 from receptor agonist to inverse agonistSHEN, Chun-Pyn; JING CHEN XIAO; ARMSTRONG, Helen et al.European journal of pharmacology. 2006, Vol 531, Num 1-3, pp 41-46, issn 0014-2999, 6 p.Article

Unravelling the complex dissociation of [³H]-rimonabant from plated CB₁ cannabinoid receptor-expressing cellsWENNERBERG, M; BALENDRAN, A; CLAPHAM, J. C et al.Fundamental & clinical pharmacology. 2010, Vol 24, Num 2, pp 181-187, issn 0767-3981, 7 p.Article

Structural and pharmacological analysis of O-2050, a putative neutral cannabinoid CB₁ receptor antagonistWILEY, Jenny L; BREIVOGEL, Christopher S; MARTIN, Billy R et al.European journal of pharmacology. 2011, Vol 651, Num 1-3, pp 96-105, issn 0014-2999, 10 p.Article

NEUROCHEMICAL BASIS OF CANNABIS ADDICTIONMALDONADO, R; BERRENDERO, F; OZAITA, A et al.Neuroscience. 2011, Vol 181, pp 1-17, issn 0306-4522, 17 p.Article

Assessment of the abuse potential of MDMA in the conditioned place preference paradigm: Role of CB1 receptorsRODRIGUEZ-ARIAS, Marta; VALVERDE, Olga; DAZA-LOSADA, Manuel et al.Progress in neuro-psychopharmacology & biological psychiatry. 2013, Vol 47, pp 77-84, issn 0278-5846, 8 p.Article

CB₁-independent mechanisms of Δ⁹-THCV, AM251 and SR141716 (rimonabant)RAFFA, R. B; WARD, S. J.Journal of clinical pharmacy and therapeutics (Print). 2012, Vol 37, Num 3, pp 260-265, issn 0269-4727, 6 p.Article

The cannabinoid CB₁ receptor is expressed on serotonergic and dopaminergic neuronsLAU, Thorsten; SCHLOSS, Patrick.European journal of pharmacology. 2008, Vol 578, Num 2-3, pp 137-141, issn 0014-2999, 5 p.Article

Effect of chronic ethanol exposure and its withdrawal on the endocannabinoid systemYARAGUDRI VINOD, K; YALAMANCHILI, Ratnakumar; SHAN XIE et al.Neurochemistry international. 2006, Vol 49, Num 6, pp 619-625, issn 0197-0186, 7 p.Article

How inverse can a neutral antagonist be? Strategic questions after the rimonabant issueGIRALDO, Jesús.Drug discovery today. 2010, Vol 15, Num 11-12, pp 411-415, issn 1359-6446, 5 p.Article

Evidence for the involvement of cannabinoid CB₁ receptors in the bimatoprost-induced contractions on the human isolated ciliary muscleROSARIA ROMANO, Maria; DIEGO LOGRANO, Marcello.Investigative ophthalmology & visual science. 2007, Vol 48, Num 8, pp 3677-3682, issn 0146-0404, 6 p.Article

Chronic use of marijuana decreases cannabinoid receptor binding and mRNA expression in the human brainVILLARES, J.Neuroscience. 2007, Vol 145, Num 1, pp 323-334, issn 0306-4522, 12 p.Article

Similar in vitro pharmacology of human cannabinoid CB₁ receptor variants expressed in CHO cellsJING CHEN XIAO; JEWELL, James P; LIN, Linus S et al.Brain research. 2008, Vol 1238, pp 36-43, issn 0006-8993, 8 p.Article

The cannabinoids R(-)-7-hydroxy-delta-6-tetra-hydrncannabinol-dimethylheptyl (HU-210), 2-O-arachidonoylglycerylether (HU-310) and arachidonyl-2-chloroethylamide (ACEA) increase isoflurane provoked sleep duration by activation of cannabinoids 1 (CB₁)-receptors in miceSCHUSTER, Johannes; ATES, Mehmet; BRUNE, Kay et al.Neuroscience letters. 2002, Vol 326, Num 3, pp 196-200, issn 0304-3940Article

Potential role of the cannabinoid receptor CB₁ in the pathogenesis of erosive and non-erosive gastro-oesophageal reflux diseaseCALABRESE, C; SPISNI, E; LIGUORI, G et al.Alimentary pharmacology & therapeutics. 2010, Vol 32, Num 4, pp 603-611, issn 0269-2813, 9 p.Article

Unique agonist-bound cannabinoid CB₁ receptor conformations indicate agonist specificity in signalingGEORGIEVA, Teodora; DEVANATHAN, Savitha; STROPOVA, Dagmar et al.European journal of pharmacology. 2008, Vol 581, Num 1-2, pp 19-29, issn 0014-2999, 11 p.Article

CB₁ receptor antagonists for the treatment of nicotine addictionCOHEN, Caroline; KODAS, Ercem; GRIEBEL, Guy et al.Pharmacology, biochemistry and behavior. 2005, Vol 81, Num 2, pp 387-395, issn 0091-3057, 9 p.Conference Paper

Multiple mechanisms of CB1 cannabinoid receptors regulationKEREN, Ora; SARNE, Yosef.Brain research. 2003, Vol 980, Num 2, pp 197-205, issn 0006-8993, 9 p.Article

Activation of the sympathetic nervous system mediates hypophagic and anxiety-like effects of CB₁ receptor blockadeBELLOCCHIO, Luigi; SORIA-GOMEZ, Edgar; VEGA, David et al.Proceedings of the National Academy of Sciences of the United States of America. 2013, Vol 110, Num 12, pp 4786-4791, issn 0027-8424, 6 p.Article

Bioactivation Pathways of the Cannabinoid Receptor 1 Antagonist RimonabantANDRESEN BERGSTRÖM, Moa; ISIN, Emre M; CASTAGNOLI, Neal et al.Drug metabolism and disposition. 2011, Vol 39, Num 10, pp 1823-1832, issn 0090-9556, 10 p.Article

Novel cannabinoid receptorsBROWN, A. J.British journal of pharmacology. 2007, Vol 152, Num 5, pp 567-575, issn 0007-1188, 9 p.Article