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Results 1 to 25 of 544

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D-Proline-based peptidomimetic inhibitors of anthrax lethal factorCALUGI, Chiara; TRABOCCHI, Andrea; LALLI, Claudia et al.European journal of medicinal chemistry. 2012, Vol 56, pp 96-107, issn 0223-5234, 12 p.Article

Metabolism of steroidal anti-inflammatory antedrugs in vitro: methyl 3,20-dioxo-11β, 17α, 21-trihydroxy-1,4-pregnadiene-16α-carboxylate; its 9a-fluorinated, and their 21-O-acyl derivativesPARK, Kwan-Kyun; KO, Dong-Hoon; ZHENGQING YOU et al.Steroids. 2003, Vol 68, Num 4, pp 315-319, issn 0039-128X, 5 p.Article

2-Arylbenzofuran-based molecules as multipotent Alzheimer's disease modifying agentsRIZZO, Stefano; TAROZZI, Andrea; ANDRISANO, Vincenza et al.European journal of medicinal chemistry. 2012, Vol 58, pp 519-532, issn 0223-5234, 14 p.Article

Application of a post-docking procedure based on MM-PBSA and MM-GBSA on single and multiple protein conformationsSGOBBA, Miriam; CAPORUSCIO, Fabiana; ANIGHORO, Andrew et al.European journal of medicinal chemistry. 2012, Vol 58, pp 431-440, issn 0223-5234, 10 p.Article

Design and Diastereoselective Synthesis of C-2,C-20-Diaryl Steroidal DerivativesREY, Jullien; O'RIORDAN, Timothy J. C; HAIPENG HU et al.European journal of organic chemistry (Print). 2012, Num 20, pp 3781-3794, issn 1434-193X, 14 p.Article

Discovery of potent inhibitors of receptor protein tyrosine phosphatase sigma through the structure-based virtual screeningPARK, Hwangseo; PHAM NGOC CHIEN; SEONG EON RYU et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 20, pp 6333-6337, issn 0960-894X, 5 p.Article

Extended targeting potential and improved synthesis of Microcin C analogs as antibacterialsVONDENHOFF, Gaston H. M; DUBILEY, Svetlana; SEVERINOV, Konstantin et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 18, pp 5462-5467, issn 0968-0896, 6 p.Article

Design of more potent squalene synthase inhibitors with multiple activitiesKOUROUNAKIS, Angeliki P; MATRALIS, Alexios N; NIKITAKIS, Anastasios et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 21, pp 7402-7412, issn 0968-0896, 11 p.Article

Synthesis and evaluation of 4-quinazolinone compounds as potential antimalarial agentsSHUREN ZHU; WANG, Joe; CHANDRASHEKAR, Gudise et al.European journal of medicinal chemistry. 2010, Vol 45, Num 9, pp 3864-3869, issn 0223-5234, 6 p.Article

Ontologies of Drug Discovery and Design for Neurology, Cardiology and OncologyVAZQUEZ-NAYA, José M; MARTINEZ-ROMERO, Marcos; PORTO-PAZOS, Ana B et al.Current pharmaceutical design (Print). 2010, Vol 16, Num 24, pp 2724-2736, issn 1381-6128, 13 p.Article

Discovery and functional evaluation of diverse novel human CB1 receptor ligandsFOLOPPE, Nicolas; BENWELL, Aren; BROOKS, Teresa D et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 15, pp 4183-4190, issn 0960-894X, 8 p.Article

Inhibition of 3(17)α-hydroxysteroid dehydrogenase (AKR1C21) by aldose reductase inhibitorsDHAGAT, Urmi; ENDO, Satoshi; HARA, Akira et al.Bioorganic & medicinal chemistry. 2008, Vol 16, Num 6, pp 3245-3254, issn 0968-0896, 10 p.Article

Carbonic anhydrases as targets for medicinal chemistrySUPURAN, Claudiu T; SCOZZAFAVA, Andrea.Bioorganic & medicinal chemistry. 2007, Vol 15, Num 13, pp 4336-4350, issn 0968-0896, 15 p.Article

Rational design of a nonpeptide general chemical scaffold for reversible inhibition of PDZ domain interactionsFUJII, Naoaki; HARESCO, Jose J; NOVAK, Kathleen A. P et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 2, pp 549-552, issn 0960-894X, 4 p.Article

Steps towards flexible docking : Modeling of three-dimensional structures of the nuclear receptors bound with peptide ligands mimicking co-activators' sequencesKURCINSKI, Mateusz; KOLINSKI, Andrzej.Journal of steroid biochemistry and molecular biology. 2007, Vol 103, Num 3-5, pp 357-360, issn 0960-0760, 4 p.Conference Paper

Brequinar derivatives and species-specific drug design for dihydroorotate dehydrogenaseHURT, Darrell E; SUTTON, Amanda E; CLARDY, Jon et al.Bioorganic & medicinal chemistry letters (Print). 2006, Vol 16, Num 6, pp 1610-1615, issn 0960-894X, 6 p.Article

Determination of hERG channel blockers using a decision treeGEPP, Michael M; HUTTER, Michael C.Bioorganic & medicinal chemistry. 2006, Vol 14, Num 15, pp 5325-5332, issn 0968-0896, 8 p.Article

Identification of chemically diverse Chk1 inhibitors by receptor-based virtual screeningFOLOPPE, Nicolas; FISHER, Lisa M; HOWES, Rob et al.Bioorganic & medicinal chemistry. 2006, Vol 14, Num 14, pp 4792-4802, issn 0968-0896, 11 p.Article

One-pot synthesis and SAR study of cis-2,6-dialkyl-4-chloro-tetrahydropyransMIRANDA, Pedro O; LEON, Leticia G; MARTIN, Victor S et al.Bioorganic & medicinal chemistry letters (Print). 2006, Vol 16, Num 12, pp 3135-3138, issn 0960-894X, 4 p.Article

Drug-herb interactions : Eliminating toxicity with hard drug designYANG, Xiao-Xia; HU, Ze-Ping; WEI DUAN et al.Current pharmaceutical design. 2006, Vol 12, Num 35, pp 4649-4664, issn 1381-6128, 16 p.Article

Design, synthesis, DNA binding, and biological activity of a series of DNA minor-groove-binding intercalating drugsBAILLY, C; POMMERY, N; HOUSSIN, R et al.Journal of pharmaceutical sciences. 1989, Vol 78, Num 11, pp 910-917, issn 0022-3549Article

Involvement of serotonin in nociceptive pathwaysROBERTS, M. H. T.Drug design and delivery. 1989, Vol 4, Num 2, pp 77-83, issn 0884-2884Article

Synthesis of mitomycin derivatives with disulfide at the 7-N side chain (3): synthesis of KW 2149 and structure-activity relationships among mitomycin derivatives with disulfide at the 7-N side chainKONO, M; SAITOH, Y; KASAI, M et al.Journal of pharmacobio-dynamics. 1989, Vol 12, Num 6, issn 0386-846X, S 138 [1 p.]Conference Paper

Fragment Based Drug Design: From Experimental to Computational ApproachesKUMAR, A; VOET, A; ZHANG, K. Y. J et al.Current medicinal chemistry. 2012, Vol 19, Num 30, pp 5128-5147, issn 0929-8673, 20 p.Conference Paper

Evaluation of structure-derived pharmacophore of soluble epoxide hydrolase inhibitors by virtual screeningMOSER, Daniel; ACHENBACH, Janosch; KLINGLER, Franca-Maria et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 21, pp 6762-6765, issn 0960-894X, 4 p.Article

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