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RDEA119/BAY 869766: A Potent, Selective, Allosteric Inhibitor of MEK1/2 for the Treatment of CancerIVERSON, Cory; LARSON, Gary; HAMATAKE, Robert et al.Cancer research (Chicago, Ill.). 2009, Vol 69, Num 17, pp 6839-6847, issn 0008-5472, 9 p.Article

ALANINE-MEDIATED REVERSIBLE INACTIVATION OF TUMOUR PYRUVATE KINASE CAUSED BY A TETRAMER-DIMER TRANSITIONSCHULZ J; SPARMANN G; HOFMANN E et al.1975; F.E.B.S. LETTERS; NETHERL.; DA. 1975; VOL. 50; NO 3; PP. 346-350; BIBL. 5REF.Article

THE ROLE OF LYSINE AND LEUCINE BINDING ON THE CATALYTICAL AND STRUCTURAL PROPERTIES OF ASPARTOKINASE III OF ESCHERICHIA COLI K12RICHAUD C; MAZAT JP; FELENBOK B et al.1974; EUROP. J. BIOCHEM.; GERM.; DA. 1974; VOL. 48; NO 1; PP. 147-156; BIBL. 35REF.Article

AROMATIC COMPOUNDS AS ALLOSTERIC INHIBITORS OF GLYCOGEN PHOSPHORYLASE BSOMAN G; PHILIP G.1974; BIOCHIM. BIOPHYS. ACTA; PAYS-BAS; DA. 1974; VOL. 358; NO 2; PP. 359-362; BIBL. 9REF.Article

THE BINDING OF REDUCED NICOTINAMIDE ADENINE DINUCLEOTIDE TO CITRATE SYNTHASE OF ESCHERICHIA COLI K12. = LA LIAISON DU NICOTINAMIDE ADENINE DINUCLEOTIDE REDUIT A LA CITRATE SYNTHASE D'E. COLI K12DUCKWORTH HW; TONG EK.1976; BIOCHEMISTRY; U.S.A.; DA. 1976; VOL. 15; NO 1; PP. 108-114; BIBL. 21 REF.Article

STRUCTURAL SPECIFICITY OF THE ALLOSTERIC INHIBITOR OF PHOSPHOENOLPYRUVATE CARBOXYLASE OF ESCHERICHIA COLI.YOSHINAGA T.1977; J. BIOCHEM.; JAP.; DA. 1977; VOL. 81; NO 3; PP. 665-671; BIBL. 17 REF.Article

A quantitative study of [3H]-D-Ala2-D-Leu5-enkephalin binding to rat brain membranes. Evidence that oxymorphone is a noncompetitive inhibitor of the lower affinity δ-binding siteROTHMAN, R. B; BOWEN, W. D; HERKENHAM, M et al.Molecular pharmacology. 1985, Vol 27, Num 3, pp 399-409, issn 0026-895XArticle

Fused thiophene derivatives as MEK inhibitorsLAING, Victoria E; BROOKINGS, Daniel C; MEIER, Christoph et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 1, pp 472-475, issn 0960-894X, 4 p.Article

INFLUENCE OF PHOSPHATE ON THE ALLOSTERIC BEHAVIOR OF YEAST PHOSPHOFRUCTOKINASE.LAURENT M; SEYDOUX F.1977; BIOCHEM. BIOPHYS. RES. COMMUNIC.; U.S.A.; DA. 1977; VOL. 78; NO 4; PP. 1289-1295; BIBL. 22 REF.Article

EFFECT OF SOME NUCLEOTIDES ON THE REGULATION OF GLYCOSAMINOGLYCAN BIOSYNTHESIS.DE LUCA G; SPEZIALE P; RINDI S et al.1976; CONNECT. TISSUE RES.; G.B.; DA. 1976; VOL. 4; NO 4; PP. 247-254; BIBL. 32 REF.Article

REGULATION OF AEROBIC FERMENTATION IN PROTOZOANS. II. ALLOSTERIC INHIBITION OF THE MALIC ENZYMEMARR JJ.1973; COMP. BIOCHEM. PHYSIOL., B; G.B.; DA. 1973; VOL. 44; NO 3; PP. 701-710; BIBL. 13 REF.Serial Issue

STOPPED FLOW FLUORESCENCE STUDIES ON THE BINDING OF REDUCED NICOTINAMIDE ADENINE DINUCLEOTIDE TO CITRATE SYNTHASE OF ESCHERICHIA COLI: EFFECTS OF PH.SADAR MH; QUEEN A; DUCKWORTH HW et al.1977; CANAD. J. BIOCHEM.; CANADA; DA. 1977; VOL. 55; NO 7; PP. 714-720; BIBL. 8 REF.Article

FLAVODOXIN: AN ALLOSTERIC INHIBITOR OF AMP NUCLEOSIDASE FROM AZOTOBACTER VINELANDII.YOSHINO M; MURAKAMI K; TSUSHIMA K et al.1976; J. BIOCHEM.; JAP.; DA. 1976; VOL. 80; NO 4; PP. 839-843; BIBL. 14 REF.Article

The role of Glu187 in the regulation of phosphofructokinase by phosphoenolpyruvateAUZAT, I; LE BRAS, G; BRANNY, P et al.Journal of molecular biology. 1994, Vol 235, Num 1, pp 68-72, issn 0022-2836Article

Crystallographic binding studies on the allosteric inhibitor glucose-6-phosphate to T state glycogen phosphorylase bJOHNSON, L. N; SNAPE, P; MARTIN, J. L et al.Journal of molecular biology. 1993, Vol 232, Num 1, pp 253-267, issn 0022-2836Article

Matrix metalloproteinase inhibitors : New challenges in the era of post broad-spectrum inhibitorsNUTI, Elisa; TUCCINARDI, Tiziano; ROSSELLO, Armando et al.Current pharmaceutical design. 2007, Vol 13, Num 20, pp 2087-2100, issn 1381-6128, 14 p.Article

Phosphoenolpyruvate-insensitive phosphofructokinase isozyme from Thermus thermophilus HB8JING XU; OSHIMA, T; YOSHIDA, M et al.Journal of biochemistry (Tokyo). 1991, Vol 109, Num 2, pp 199-203, issn 0021-924X, 5 p.Article

Preclinical Characterization of BMS-791325, an Allosteric Inhibitor of Hepatitis C Virus NS5B PolymeraseLEMM, Julie A; MENGPING LIU; KNIPE, Jay O et al.Antimicrobial agents and chemotherapy. 2014, Vol 58, Num 6, pp 3485-3495, issn 0066-4804, 11 p.Article

Receptor binding mode and pharmacological characterization of a potent and selective dual CXCR1/CXCR2 non-competitive allosteric inhibitorBERTINI, R; BARCELOS, L. S; CORSI, M. M et al.British journal of pharmacology. 2012, Vol 165, Num 2, pp 436-454, issn 0007-1188, 19 p.Article

New Directions in Targeting Protein Kinases: Focusing Upon True Allosteric and Bivalent InhibitorsLAMBA, Vandana; GHOSH, Indraneel.Current pharmaceutical design (Print). 2012, Vol 18, Num 20, pp 2936-2945, issn 1381-6128, 10 p.Article

A general technique to rank protein-ligand binding affinities and determine allosteric versus direct binding site competition in compound mixturesANNIS, D. Allen; NAZEF, Naim; CHUANG, Cheng-Chi et al.Journal of the American Chemical Society. 2004, Vol 126, Num 47, pp 15495-15503, issn 0002-7863, 9 p.Article

Inhibition of hepatic tryptophan-2,3-dioxygenase : Superior potency of melatonin over serotoninWALSH, H. A; DAYA, S.Journal of pineal research. 1997, Vol 23, Num 1, pp 20-23, issn 0742-3098Article

Enhanced oxygenation in vivo by allosteric inhibitors of hemoglobin saturationKHANDELWAL, S. R; RANDAD, R. S; PECK-SUN LIN et al.American journal of physiology. Heart and circulatory physiology. 1993, Vol 34, Num 4, pp H1450-H1453, issn 0363-6135Article

Characterization of pyridoxal 5'-phosphate affinity labeling of band 3 protein: evidence for allosterically interacting transport inhibitory subdomainsSALHANY, J. M; RAUENBUEHLER, P. B; SLOAN, R. L et al.The Journal of biological chemistry (Print). 1987, Vol 262, Num 33, pp 15965-15973, issn 0021-9258Article

Phosphorylase a is an allosteric inhibitor of the glycogen and microsomal forms of rat hepatic protein phosphatase-1ALEMANY, S; COHEN, P.FEBS letters. 1986, Vol 198, Num 2, pp 194-202, issn 0014-5793Article

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