Nonsteroidal Selective Androgen Receptor Modulators (SARMs): Dissociating the Anabolic and Androgenic Activities of the Androgen Receptor for Therapeutic BenefitMOHLER, Michael L; BOHL, Casey E; JONES, Amanda et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 12, pp 3597-3617, issn 0022-2623, 21 p.Article

Mass spectrometry of hydantoin-derived selective androgen receptor modulatorsTHEVIS, Mario; KOHLER, Maxie; SCHLÖRER, Nils et al.Journal of mass spectrometry. 2008, Vol 43, Num 5, pp 639-650, issn 1076-5174, 12 p.Article

Design, Synthesis, and Biological Evaluation of 16-Substituted 4-Azasteroids as Tissue-Selective Androgen Receptor Modulators (SARMs)MITCHELL, Helen J; DANKULICH, William P; LEU, Chih-Tai et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 15, pp 4578-4581, issn 0022-2623, 4 p.Article

Synthesis of potent, substituted carbazoles as selective androgen receptor modulators (SARMs)MILLER, Chris P; BHAKET, Pushpal; MUTHUKAMAN, Nagarajan et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 24, pp 7516-7520, issn 0960-894X, 5 p.Article

Novel series of potent, nonsteroidal, selective androgen receptor modulators based on 7H-[1,4 ]oxazino [3,2 -g]quinolin -7 -onesHIGUCHI, Robert I; ARIENTI, Kristen L; SCHRADER, William T et al.Journal of medicinal chemistry (Print). 2007, Vol 50, Num 10, pp 2486-2496, issn 0022-2623, 11 p.Article

Discovery of a novel series of nonsteroidal androgen receptor modulators : 5-or 6-oxachrysen-2-onesSHUO ZHAO; YIXING SHEN; VAN OEVEREN, Arjan et al.Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 11, pp 3431-3435, issn 0960-894X, 5 p.Article

Mass spectrometry of selective androgen receptor modulatorsTHEVIS, Mario; SCHÄNZER, Wilhelm.Journal of mass spectrometry. 2008, Vol 43, Num 7, pp 865-876, issn 1076-5174, 12 p.Article

Potent anti-prostate cancer agents derived from a novel androgen receptor down-regulating agentPURUSHOTTAMACHAR, Puranik; KHANDELWAL, Aakanksha; VASAITIS, Tadas S et al.Bioorganic & medicinal chemistry. 2008, Vol 16, Num 7, pp 3519-3529, issn 0968-0896, 11 p.Article

Targeted intracellular protein degradation induced by a small molecule : En route to chemical proteomicsSCHNEEKLOTH, Ashley R; PUCHEAULT, Mathieu; HYUN SEOP TAE et al.Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 22, pp 5904-5908, issn 0960-894X, 5 p.Article

Discovery of an androgen receptor modulator pharmacophore based on 2-quinolinonesVAN OEVEREN, Arjan; PIO, Barbara A; TEGLEY, Christopher M et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 6, pp 1523-1526, issn 0960-894X, 4 p.Article

Substituted 6 -(1 -Pyrrolidine )quinolin -2(1H)-ones as Novel Selective Androgen Receptor ModulatorsMARTINBOROUGH, Esther; YIXING SHEN; HUMBERTO VIVEROS, O et al.Journal of medicinal chemistry (Print). 2007, Vol 50, Num 21, pp 5049-5052, issn 0022-2623, 4 p.Article

Discovery of potent and muscle selective androgen receptor modulators through scaffold modificationsLI, James J; SUTTON, James C; GOLLA, Rajasree et al.Journal of medicinal chemistry (Print). 2007, Vol 50, Num 13, pp 3015-3025, issn 0022-2623, 11 p.Article

Discovery of potent, orally-active, and muscle-selective androgen receptor modulators based on an N-aryl-hydroxybicyclohydantoin scaffoldCHONGQING SUN; ROBL, Jeffrey A; FURA, Aberra et al.Journal of medicinal chemistry (Print). 2006, Vol 49, Num 26, pp 7596-7599, issn 0022-2623, 4 p.Article

Tetrahydroquinolines as a novel series of nonsteroidal selective androgen receptor modulators: Structural requirements for better physicochemical and biological propertiesNAGATA, Naoya; MIYAKAWA, Motonori; AMANO, Seiji et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 21, pp 6310-6313, issn 0960-894X, 4 p.Article

Novel selective androgen receptor modulators : SAR studies on 6-bisalkylamino-2-quinolinonesVAN OEVEREN, Arjan; MOTAMEDI, Mehrnoush; NEGRO-VILAR, Andrés et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 6, pp 1527-1531, issn 0960-894X, 5 p.Article

Synthesis and SAR of novel hydantoin derivatives as selective androgen receptor modulatorsXUQING ZHANG; ALLAN, George F; SBRISCIA, Tifanie et al.Bioorganic & medicinal chemistry letters (Print). 2006, Vol 16, Num 22, pp 5763-5766, issn 0960-894X, 4 p.Article

N-Aryl-oxazolidin-2-imine Muscle Selective Androgen Receptor Modulators Enhance Potency through Pharmacophore ReorientationNIRSCHL, Alexandra A; YAN ZOU; BEEHLER, Blake C et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 9, pp 2794-2798, issn 0022-2623, 5 p.Article

Synthesis of potent and tissue-selective androgen receptor modulators (SARMs): 2-(2,2,2)-trifluoroethyl-benzimidazole scaffoldNG, Raymond A; LANTER, James C; ALFORD, Vernon C et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 6, pp 1784-1787, issn 0960-894X, 4 p.Article

Serendipitous discovery of novel imidazolopyrazole scaffold as selective androgen receptor modulatorsXUQING ZHANG; XIAOJIE LI; ALLAN, George F et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 2, pp 439-443, issn 0960-894X, 5 p.Article

Effect of B-ring substitution pattern on binding mode of propionamide selective androgen receptor modulatorsBOHL, Casey E; ZENGRU WU; JIYUN CHEN et al.Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 20, pp 5567-5570, issn 0960-894X, 4 p.Article

Tandem optimization of target activity and elimination of mutagenic potential in a potent series of N-aryl bicyclic hydantoin-based selective androgen receptor modulatorsHAMANN, Lawrence G; MANFREDI, Mark C; FURA, Aberra et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 7, pp 1860-1864, issn 0960-894X, 5 p.Article

Synthesis and SAR of tetrahydropyrrolo[1,2 -b] [1,2,5]thiadiazol -2 (3H) -one 1,1-dioxide analogues as highly potent selective androgen receptor modulatorsMANFREDI, Mark C; YINGZHI BI; HAMANN, Lawrence G et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 16, pp 4487-4490, issn 0960-894X, 4 p.Article

Design and synthesis of tricyclic tetrahydroquinolines as a new series of nonsteroidal selective androgen receptor modulators (SARMs)NAGATA, Naoya; MIYAKAWA, Motonori; AMANO, Seiji et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 6, pp 1744-1747, issn 0960-894X, 4 p.Article

Emerging drugs : mechanism of action, mass spectrometry and doping control analysisTHEVIS, Mario; THOMAS, Andreas; KOHLER, Maxie et al.Journal of mass spectrometry. 2009, Vol 44, Num 4, pp 442-460, issn 1076-5174, 19 p.Article

Synthesis, Structure—Activity Relationships, and Characterization of Novel Nonsteroidal and Selective Androgen Receptor ModulatorsSCHLIENGER, Nathalie; LUND, Birgitte W; GARDELL, Luis R et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 22, pp 7186-7191, issn 0022-2623, 6 p.Article