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Synthesis of Kalasinamide, a Putative Plant Defense PhototoxinGANDY, Michael N; PIGGOTT, Matthew J.Journal of natural products (Print). 2008, Vol 71, Num 5, pp 866-868, issn 0163-3864, 3 p.Article

Synthesis of 6-substituted 9-methoxy-11H-indeno[1,2-c]quinoline-11-one derivatives as potential anticancer agentsTSENG, Chih-Hua; CHEN, Yeh-Long; YANG, Chiao-Li et al.Bioorganic & medicinal chemistry. 2012, Vol 20, Num 14, pp 4397-4404, issn 0968-0896, 8 p.Article

Synthesis and biological evaluation of novel N-acyl substituted quinolin-2(1H)-one derivatives as potential antimicrobial agentsLIU, Hong-Bin; HUI TANG; DAN YANG et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 18, pp 5845-5848, issn 0960-894X, 4 p.Article

N.M.R. spectral studies of some quinolone derivatives. VIII: 13C - 1H coupling constants for the 2-quinolone systemOSBORNE, A. G.Spectroscopy letters. 1994, Vol 27, Num 1, pp 1-22, issn 0038-7010Article

The 'pyrono route' to 4-hydroxy-2-quinolones and 4-hydroxy-2-pyridonesKAPPE, T.Il Farmaco (Pavia). 1999, Vol 54, Num 5, pp 309-315, issn 0014-827XArticle

Electron ionization-induced fragmentation of N- and O-alkoxymethylated carbostyril and phenanthridinoneSZMIGIELSKI, Rafat; DANIKIEWICZ, Witold.Journal of mass spectrometry. 2004, Vol 39, Num 7, pp 781-790, issn 1076-5174, 10 p.Article

Intramolecular Aldol Reaction of N-Acylated (2-Aminophenyl)-α-oxoacetic Acids: Rapid Access to Tri- and Tetracyclic 1,2-Dihydroquinolin-2(1H)-onesHELLAL, Malik; CUNY, Gregory D.Journal of organic chemistry. 2010, Vol 75, Num 10, pp 3465-3468, issn 0022-3263, 4 p.Article

Palladium-Catalyzed Intramolecular Amidation of C(sp2)-H Bonds: Synthesis of 4-Aryl-2-quinolinonesINAMOTO, Kiyofumi; SAITO, Tadataka; HIROYA, Kou et al.Journal of organic chemistry. 2010, Vol 75, Num 11, pp 3900-3903, issn 0022-3263, 4 p.Article

Synthesis and SAR studies of 2-oxoquinoline derivatives as CB2 receptor inverse agonistsRAITIO, Katri H; SAVINAINEN, Juha R; VEPSÄLÄINEN, Jouko et al.Journal of medicinal chemistry (Print). 2006, Vol 49, Num 6, pp 2022-2027, issn 0022-2623, 6 p.Article

Carbamates as potent calcitonin gene-related peptide antagonists with improved solution stabilityDEGNAN, Andrew P; CONWAY, Charles M; DALTERIO, Richard A et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 13, pp 3555-3558, issn 0960-894X, 4 p.Article

Pyrrolo[3,4-h]quinolinones a new class of photochemotherapeutic agentsBARRAJA, Paola; DIANA, Patrizia; MONTALBANO, Alessandra et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 7, pp 2326-2341, issn 0968-0896, 16 p.Article

Farnesyltransferase Inhibitors : A Detailed Chemical View on an Elusive Biological ProblemSOUSA, Sérgio F; FERNANDES, Pedro A; RAMOS, Maria Joao et al.Current medicinal chemistry. 2008, Vol 15, Num 15, pp 1478-1492, issn 0929-8673, 15 p.Article

Fluorescent retinoid X receptor ligands for fluorescence polarization assayYAMADA, Shoya; OHSAWA, Fuminori; FUJII, Shuji et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 17, pp 5143-5146, issn 0960-894X, 4 p.Article

Multivariate SAR/QSAR of 3-aryl-4-hydroxyquinolin-2(1H)-one derivatives as type I fatty acid synthase (FAS) inhibitorsBORGES DE MELO, Eduardo.European journal of medicinal chemistry. 2010, Vol 45, Num 12, pp 5817-5826, issn 0223-5234, 10 p.Article

Effect of TA-270. a novel quinolinone derivative, on antigen-induced nasal blockage in a guinea pig model of allergic rhinitisMIZUTANI, Nobuaki; AOKI, Yasuo; NABE, Takeshi et al.European journal of pharmacology. 2009, Vol 602, Num 1, pp 138-142, issn 0014-2999, 5 p.Article

Selective Synthesis of 3-Aryl Quinolin-2(1H)-ones and 3-(1-Arylmethylene)oxindoles Involving a 2-Fold Arene C-H Activation ProcessTANG, Dong-Jun; TANG, Bo-Xiao; LI, Jin-Heng et al.Journal of organic chemistry. 2009, Vol 74, Num 17, pp 6749-6755, issn 0022-3263, 7 p.Article

Impact on famesyltransferase inhibition of 4-chlorophenyl moiety replacement in the Zamestra® seriesANGIBAUD, Patrick; MEVELLEC, Laurence; VAN DUN, Jacky et al.European journal of medicinal chemistry. 2007, Vol 42, Num 5, pp 702-714, issn 0223-5234, 13 p.Article

Diels-Alder reactions of nitro-2(1H)-pyridones with 2,3-dimethyl-1,3-butadieneFUJITA, Reiko; WATANABE, Kazuhiro; NISHIUCHI, Yasuhiro et al.Chemical and pharmaceutical bulletin. 2001, Vol 49, Num 5, pp 601-605, issn 0009-2363Article

Discovery of substituted phenyl urea derivatives as novel long-acting β2-adrenoreceptor agonistsPEREZ, Daniel; CRESPO, Maribel; PUIG, Carles et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 5, pp 1545-1548, issn 0960-894X, 4 p.Article

Synthesis of 3-0-methylviridicatin analogues with improved anti-TNF-a propertiesRIBEIRO, Nigel; TABAKA, Helena; PELUSO, Jean et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 20, pp 5523-5524, issn 0960-894X, 2 p.Article

Synthetic study on the unique dimeric arylpiperazine: Access to the minor contaminant of AripiprazoleTORISAWA, Yasuhiro; SHINHAMA, Koichi; NISHI, Takao et al.Bioorganic & medicinal chemistry letters (Print). 2003, Vol 13, Num 1, pp 65-68, issn 0960-894X, 4 p.Article

Synthesis of phenanthridones using diels-alder reactions of 4-substituted 2(1H)-quinolones acting as dienophilesFUJITA, Reiko; WATANABE, Kazuhiro; YOSHISUJI, Toshiteru et al.Chemical and pharmaceutical bulletin. 2001, Vol 49, Num 4, pp 407-412, issn 0009-2363Article

Evaluation and biological properties of reactive ligands for the mapping of the glycine site on the N-methyl-D-aspartate (NMDA) receptorKREIMEYER, A; LAUBE, B; STURGESS, M et al.Journal of medicinal chemistry (Print). 1999, Vol 42, Num 21, pp 4394-4404, issn 0022-2623Article

Proton exchange reactions in isotope chemistry (I)ZHIGANG JIAN; RAY, Tapan; WU, Amy et al.Journal of labelled compounds & radiopharmaceuticals. 2012, Vol 55, Num 1-2, pp 84-87, issn 0362-4803, 4 p.Article

Facile synthesis of 4-acetyl-coumarins, -thiocoumarin and -quinolin-2(1H)-one via very high α-regioselective Heck coupling on tosylatesVALENTE, Sergio; KIRSCH, Gilbert.Tetrahedron letters. 2011, Vol 52, Num 27, issn 0040-4039, 3406, 3429-3432 [5 p.]Article

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