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A PHASE IIA RANDOMIZED, PLACEBO-CONTROLLED CLINICAL TRIAL TO STUDY THE EFFICACY AND SAFETY OF THE SELECTIVE ANDROGEN RECEPTOR MODULATOR (SARM), MK-0773 IN FEMALE PARTICIPANTS WITH SARCOPENIAPAPANICOLAOU, D. A; ATHER, S. N; ZHU, H et al.The Journal of nutrition, health & aging. 2013, Vol 17, Num 6, pp 533-543, issn 1279-7707, 11 p.Article

Enhanced evaluation of selective androgen receptor modulators in vivoOTTO-DUESSEL, M; HE, M; ADAMSON, T. W et al.Andrology (Print). 2013, Vol 1, Num 1, pp 29-36, issn 2047-2919, 8 p.Article

Nonsteroidal Selective Androgen Receptor Modulators (SARMs): Dissociating the Anabolic and Androgenic Activities of the Androgen Receptor for Therapeutic BenefitMOHLER, Michael L; BOHL, Casey E; JONES, Amanda et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 12, pp 3597-3617, issn 0022-2623, 21 p.Article

Bone anabolic effects of S-40503, a novel nonsteroidal selective androgen receptor modulator (SARM), in rat models of osteoporosisHANADA, Keigo; FURUYA, Kazuyuki; YAMAMOTO, Noriko et al.Biological & pharmaceutical bulletin. 2003, Vol 26, Num 11, pp 1563-1569, issn 0918-6158, 7 p.Article

17β-Hydroxyestra-4,9,11-trien-3-one (trenbolone) exhibits tissue selective anabolic activity: effects on muscle, bone, adiposity, hemoglobin, and prostateYARROW, Joshua F; CONOVER, Christine F; PINGEL, Jennifer E et al.American journal of physiology. Endocrinology and metabolism. 2011, Vol 63, Num 4, issn 0193-1849, E650-E660Article

Combination Treatment With a Selective Androgen Receptor Modulator (SARM) and a Bisphosphonate Has Additive Effects in Osteopenic Female RatsVAJDA, Eric G; HOGUE, Aimee; VAN OEVEREN, Arjan et al.Journal of bone and mineral research (Print). 2009, Vol 24, Num 2, pp 231-240, issn 0884-0431, 10 p.Article

Mass spectrometry of hydantoin-derived selective androgen receptor modulatorsTHEVIS, Mario; KOHLER, Maxie; SCHLÖRER, Nils et al.Journal of mass spectrometry. 2008, Vol 43, Num 5, pp 639-650, issn 1076-5174, 12 p.Article

A selective androgen receptor modulator with minimal prostate hypertrophic activity restores lean body mass in aged orchidectomized male ratsALLAN, George; SBRISCIA, Tifanie; LINTON, Olivia et al.Journal of steroid biochemistry and molecular biology. 2008, Vol 110, Num 3-5, pp 207-213, issn 0960-0760, 7 p.Article

Androgen receptor as a therapeutic targetWENQING GAO.Advanced drug delivery reviews. 2010, Vol 62, Num 13, pp 1277-1284, issn 0169-409X, 8 p.Article

Synthesis and SAR of tetrahydropyrrolo[1,2 -b] [1,2,5]thiadiazol -2 (3H) -one 1,1-dioxide analogues as highly potent selective androgen receptor modulatorsMANFREDI, Mark C; YINGZHI BI; HAMANN, Lawrence G et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 16, pp 4487-4490, issn 0960-894X, 4 p.Article

Anti-Androgenic Effects of S-40542, A Novel Non-Steroidal Selective Androgen Receptor Modulator (SARM) for the Treatment of Benign Prostatic HyperplasiaNEJISHIMA, Hiroaki; YAMAMOTO, Noriko; SUZUKI, Mika et al.The Prostate. 2012, Vol 72, Num 14, pp 1580-1587, issn 0270-4137, 8 p.Article

Mass spectrometry of selective androgen receptor modulatorsTHEVIS, Mario; SCHÄNZER, Wilhelm.Journal of mass spectrometry. 2008, Vol 43, Num 7, pp 865-876, issn 1076-5174, 12 p.Article

Synthesis of potent, substituted carbazoles as selective androgen receptor modulators (SARMs)MILLER, Chris P; BHAKET, Pushpal; MUTHUKAMAN, Nagarajan et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 24, pp 7516-7520, issn 0960-894X, 5 p.Article

Novel series of potent, nonsteroidal, selective androgen receptor modulators based on 7H-[1,4 ]oxazino [3,2 -g]quinolin -7 -onesHIGUCHI, Robert I; ARIENTI, Kristen L; SCHRADER, William T et al.Journal of medicinal chemistry (Print). 2007, Vol 50, Num 10, pp 2486-2496, issn 0022-2623, 11 p.Article

Discovery of a novel series of nonsteroidal androgen receptor modulators : 5-or 6-oxachrysen-2-onesSHUO ZHAO; YIXING SHEN; VAN OEVEREN, Arjan et al.Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 11, pp 3431-3435, issn 0960-894X, 5 p.Article

Pharmacokinetics and pharmacodynamics of nonsteroidal androgen receptor ligandsWENQING GAO; KIM, Juhyun; DALTON, James T et al.Pharmaceutical research. 2006, Vol 23, Num 8, pp 1641-1658, issn 0724-8741, 18 p.Article

Design, Synthesis, and Biological Evaluation of 16-Substituted 4-Azasteroids as Tissue-Selective Androgen Receptor Modulators (SARMs)MITCHELL, Helen J; DANKULICH, William P; LEU, Chih-Tai et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 15, pp 4578-4581, issn 0022-2623, 4 p.Article

Selective androgen receptor modulators: in vitro and in vivo metabolism and analysisDE RIJKE, Eva; ESSERS, Martien L; RIJK, Jeroen C. W et al.Food additives & contaminants. Part A. Chemistry, analysis, control, exposure & risk assessment (Print). 2013, Vol 30, Num 9, pp 1517-1526, issn 1944-0049, 10 p.Article

Substituted 6 -(1 -Pyrrolidine )quinolin -2(1H)-ones as Novel Selective Androgen Receptor ModulatorsMARTINBOROUGH, Esther; YIXING SHEN; HUMBERTO VIVEROS, O et al.Journal of medicinal chemistry (Print). 2007, Vol 50, Num 21, pp 5049-5052, issn 0022-2623, 4 p.Article

Potent anti-prostate cancer agents derived from a novel androgen receptor down-regulating agentPURUSHOTTAMACHAR, Puranik; KHANDELWAL, Aakanksha; VASAITIS, Tadas S et al.Bioorganic & medicinal chemistry. 2008, Vol 16, Num 7, pp 3519-3529, issn 0968-0896, 11 p.Article

Targeted intracellular protein degradation induced by a small molecule : En route to chemical proteomicsSCHNEEKLOTH, Ashley R; PUCHEAULT, Mathieu; HYUN SEOP TAE et al.Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 22, pp 5904-5908, issn 0960-894X, 5 p.Article

Discovery of an androgen receptor modulator pharmacophore based on 2-quinolinonesVAN OEVEREN, Arjan; PIO, Barbara A; TEGLEY, Christopher M et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 6, pp 1523-1526, issn 0960-894X, 4 p.Article

A selective androgen receptor modulator that reduces prostate tumor size and prevents orchidectomy-induced bone loss in ratsALLAN, George; LAI, Muh-Tsann; LUNDEEN, Scott et al.Journal of steroid biochemistry and molecular biology. 2007, Vol 103, Num 1, pp 76-83, issn 0960-0760, 8 p.Article

Discovery of potent, orally-active, and muscle-selective androgen receptor modulators based on an N-aryl-hydroxybicyclohydantoin scaffoldCHONGQING SUN; ROBL, Jeffrey A; FURA, Aberra et al.Journal of medicinal chemistry (Print). 2006, Vol 49, Num 26, pp 7596-7599, issn 0022-2623, 4 p.Article